SCHEMBL2485723

SCHEMBL2485723

CC(C)(NC(=O)C1CCC1)C(=O)Nc1nc(-c2ccc(F)cc2)c(Oc2ccc(F)cc2)s1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACHE P22303 8/20 0.45
ALDH1A1 P00352 2/20 0.41
PKM P14618 1/20 0.41
HTT P42858 1/20 0.40
RORC P51449 2/20 0.38
ABL1 P00519 3/20 0.38
MAPT P10636 1/20 0.38
GSK3B P49841 1/20 0.37
MAPK14 Q16539 1/20 0.37
CSNK1D P48730 1/20 0.37
CSNK1E P49674 1/20 0.37
SCN9A Q15858 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2487464 0.92 ACHE (0.44) ACHEALDH1A1PKMHTTRORC
SCHEMBL12206938 0.87 ACHE (0.36) ACHEALDH1A1PKMHTTABL1
SCHEMBL2313625 0.87 CSNK1D (0.39) ACHEALDH1A1PKMHTTRORC
SCHEMBL2321338 0.86 ACHE (0.39) ACHEALDH1A1PKMHTTRORC
SCHEMBL2487593 0.85 ALDH1A1 (0.46) ACHEALDH1A1PKMHTTRORC
SCHEMBL2314979 0.85 ALDH1A1 (0.41) ACHEALDH1A1PKMHTTRORC
SCHEMBL2490939 0.85 RORC (0.41) ACHEALDH1A1PKMHTTRORC
SCHEMBL2484976 0.84 ALDH1A1 (0.45) ACHEALDH1A1PKMHTTRORC
SCHEMBL2485003 0.84 RORC (0.42) ACHEALDH1A1PKMHTTRORC
SCHEMBL2490686 0.84 SMN1; SMN2 (0.45) ALDH1A1PKMRORCMAPTPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2380631-A1 Heteroaryl derivatives as DGAT1 inhibitors Novartis AG (CH) 2011-10-26 EP disclosed