SCHEMBL24858675

SCHEMBL24858675

O=C(c1ccc(F)nc1)c1ccc2c(c1)c(F)nn2PI

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
KCNQ3 O43525 1/20 0.32
KCNQ2 O43526 1/20 0.32
SPR P35270 1/20 0.31
EPHX2 P34913 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24858683 0.82 MAPK1 (0.37) NPC1
SCHEMBL24858305 0.78 CCNB2 (0.31)
SCHEMBL31195590 0.73 SPR (0.43) SPR
SCHEMBL34460387 0.73 SPR (0.43) SPR
SCHEMBL27594193 0.72 RXFP1 (0.53) NPC1RXFP1KCNQ3KCNQ2EPHX2
SCHEMBL24858674 0.71 CYP4F2 (0.39) NPC1
SCHEMBL5046191 0.66 NPC1 (0.66) NPC1RXFP1KCNQ3KCNQ2
SCHEMBL5042391 0.64 ALDH1A1 (0.54) NPC1RXFP1EPHX2
SCHEMBL23559727 0.64 KDM4E (0.43)
SCHEMBL25015127 0.63 KDM4E (0.41) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023272410-A1 ERα RECEPTOR COVALENT BINDING ANTAGONIST 北京盛诺基医药科技股份有限公司 2023-01-05 WO disclosed