SCHEMBL24858683

SCHEMBL24858683

O=C(c1ccc(Cl)cc1)c1ccc2c(c1)c(F)nn2PI

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.37
SRD5A2 P31213 1/20 0.37
HDAC3 O15379 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC2 Q92769 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
HPGD P15428 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
HTT P42858 3/20 0.33
AKR1C3 P42330 2/20 0.33
AKR1C2 P52895 2/20 0.33
VNN1 O95497 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
HSD17B1 P14061 1/20 0.33
HSD17B2 P37059 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24858305 0.88 CCNB2 (0.31)
SCHEMBL24858675 0.82 NPC1 (0.33) NPC1
SCHEMBL24858713 0.74 HDAC8 (0.41) MAPK1SRD5A2HDAC3HDAC1HDAC2
SCHEMBL24858681 0.70 DGAT2 (0.37) CNR1CNR2
SCHEMBL23559727 0.66 KDM4E (0.43) HPGDHTTTSHRHSD17B10TDP1
SCHEMBL25015127 0.65 KDM4E (0.41) NPC1SMN1; SMN2KMT2ACYP2D6HSD17B10
SCHEMBL10697158 0.64 SRD5A2 (0.80) MAPK1SRD5A2HPGDCNR1CNR2
SCHEMBL51827 0.64 SRD5A2 (0.80) MAPK1SRD5A2HPGDCNR1CNR2
SCHEMBL9065412 0.64 SRD5A2 (0.80) MAPK1SRD5A2HPGDCNR1CNR2
SCHEMBL1681512 0.64 SRD5A2 (0.80) MAPK1SRD5A2HPGDCNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023272410-A1 ERα RECEPTOR COVALENT BINDING ANTAGONIST 北京盛诺基医药科技股份有限公司 2023-01-05 WO disclosed