SCHEMBL24858713

SCHEMBL24858713

O=C(c1ccc(Cl)cc1)c1ccc2c(cnn2PI)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
KMO O15229 2/20 0.39
MAPK1 P28482 2/20 0.39
SRD5A2 P31213 1/20 0.39
HTT P42858 2/20 0.38
MAOB P27338 3/20 0.37
MAOA P21397 2/20 0.37
HPGD P15428 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
ACHE P22303 1/20 0.37
VNN1 O95497 2/20 0.36
USP2 O75604 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24858413 0.86 HSD17B1 (0.37) KMOMAOBMAOAHPGDACHE
SCHEMBL24858683 0.74 MAPK1 (0.37) HDAC8HDAC3HDAC1HDAC2HDAC6
SCHEMBL5518679 0.70 SRD5A2 (0.61) MAPK1SRD5A2HTTHPGDNPC1
SCHEMBL21538290 0.69 DEGS1 (0.49) HTTNPC1RAB9ALMNACYP1A2
SCHEMBL24858672 0.69 RXRA (0.56) HDAC8HDAC3HDAC1HDAC2HDAC6
SCHEMBL9475353 0.69 SRD5A2 (0.59) MAPK1SRD5A2HTTHPGDNPC1
SCHEMBL19772304 0.68 SLC22A12 (0.40) HDAC8KMONPC1RAB9ACYP1A2
SCHEMBL20176165 0.68 HDAC8 (0.39) HDAC8KMOMAPTKMT2A
SCHEMBL24858407 0.68 CA1 (0.38)
SCHEMBL8967726 0.67 SRD5A2 (0.57) MAPK1SRD5A2HTTHPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023272410-A1 ERα RECEPTOR COVALENT BINDING ANTAGONIST 北京盛诺基医药科技股份有限公司 2023-01-05 WO disclosed