SCHEMBL248669

SCHEMBL248669

O=C(Cl)c1cccc(OC(F)(F)F)c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KAT6A Q92794 4/20 0.51
MGLL Q99685 1/20 0.49
TAS1R3 Q7RTX0 1/20 0.49
TAS1R1 Q7RTX1 1/20 0.49
TAS1R2 Q8TE23 1/20 0.49
HDAC8 Q9BY41 1/20 0.47
HSD11B1 P28845 1/20 0.47
MAOB P27338 1/20 0.46
MRGPRX4 Q96LA9 2/20 0.46
GPR139 Q6DWJ6 1/20 0.45
P2RX1 P51575 1/20 0.45
DDR1 Q08345 1/20 0.44
NAMPT P43490 1/20 0.44
MAPK14 Q16539 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29461392 1.00 KAT6A (0.51) KAT6AMGLLTAS1R3TAS1R1TAS1R2
SCHEMBL10912843 0.88 ABL1 (0.42) KAT6AMGLLTAS1R3TAS1R1TAS1R2
SCHEMBL10562151 0.86 KAT6A (0.40) KAT6AMGLLTAS1R3TAS1R1TAS1R2
SCHEMBL2107071 0.86 NPC1 (0.58) P2RX1
SCHEMBL690501 0.85 KAT6A (0.54) KAT6AMGLLTAS1R3TAS1R1TAS1R2
SCHEMBL5866992 0.85 MAPT (0.49) KAT6A
SCHEMBL27971413 0.84 KAT6A (0.50) KAT6AMGLLTAS1R3TAS1R1TAS1R2
Benzoyl Chloride SCHEMBL8173899 0.84 KAT6A (0.48) KAT6AMGLLTAS1R3TAS1R1TAS1R2
SCHEMBL11023974 0.84 ALDH1A1 (0.43) KAT6AMGLLHDAC8MRGPRX4
SCHEMBL29459930 0.84 MRGPRX4 (0.61) KAT6ATAS1R3TAS1R1TAS1R2MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 405 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117105826-A HNO-releasable compound and preparation method thereof 海南大学 2023-11-24 CN claimed
CN-117105897-A HNO donor compound and preparation method thereof 海南大学 2023-11-24 CN claimed
CN-114230495-B Hydrogenated nitrosyl donor and preparation method thereof 海南大学 2023-01-06 CN claimed
CN-114230495-A Hydrogenated nitrosyl donor and preparation method thereof 海南大学 2022-03-25 CN claimed
CN-114195731-A Hydrogenated nitrosyl donor compound and preparation method thereof 海南大学 2022-03-18 CN claimed
US-20250248990-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2025-08-07 US disclosed
US-20250243177-A1 sGC STIMULATORS CYCLERION THERAPEUTICS, INC. 2025-07-31 US disclosed
US-12144806-B2 Quinolines that modulate SERCA and their use for treating disease NEURODON CORPORATION (US) 2024-11-19 US disclosed
US-20240277694-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2024-08-22 US disclosed
CN-118221613-A Substituted piperazine compound and medical application thereof 中国人民解放军军事科学院军事医学研究院 2024-06-21 CN disclosed
US-11992487-B2 Quinolines that modulate SERCA and their use for treating disease NEURODON CORPORATION (US) 2024-05-28 US disclosed
EP-4037685-B9 QUINOLINE THAT MODULATE SERCA AND ITS USE FOR TREATING DISEASE NEURODON CORP (US) 2024-03-06 EP disclosed
US-5221685-A Insecticides, miticides or fungicides UBE INDUSTRIES, LTD. (JP) 1993-06-22 US disclosed
EP-0497367-A1 Thiazoline derivatives, processes for their preparation and pesticidal compositions containing them UBE INDUSTRIES, LTD. (JP) 1992-08-05 EP disclosed
EP-0124002-B1 PROCESS FOR THE PREPARATION OF AROMATIC COMPOUNDS CONTAINING PERFLUORINATED SIDE CHAINS LINKED BY A HETEROATOM BAYER AG (DE) 1986-11-12 EP disclosed
US-4600787-A Process for the preparation of aromatic compounds which contain perfluorinated side-chains bonded via a heteroatom BAYER AKTIENGESELLSCHAFT (DE) 1986-07-15 US disclosed
EP-0124002-A1 Process for the preparation of aromatic compounds containing perfluorinated side chains linked by a heteroatom BAYER AG (DE) 1984-11-07 EP disclosed
US-4348395-A 1,4-Dihydropyridazine compounds BAYER AKTIENGESELLSCHAFT (DE) 1982-09-07 US disclosed
EP-0001439-B1 1-N-SUBSTITUTED 1.4-DIHYDROPYRIDAZINE DERIVATIVES, METHOD FOR THEIR PREPARATION AND THEIR USE FOR PHARMACEUTICALS BAYER AG (DE) 1981-01-28 EP disclosed
EP-0001439-A1 1-N-substituted 1.4-dihydropyridazine derivatives, method for their preparation and their use for pharmaceuticals BAYER AG (DE) 1979-04-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11992487-B2 Quinolines that modulate SERCA and their use for treating disease ATP2A1, ATP2A3, ATP2A2 KAT6A 3520/4885MGLL 2015/4885TAS1R3 3383/4885
US-12144806-B2 Quinolines that modulate SERCA and their use for treating disease ATP2A1, ATP2A3, ATP2A2 KAT6A 3520/4885MGLL 2015/4885TAS1R3 3383/4885
US-20250248990-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 KAT6A 3520/4885MGLL 2015/4885TAS1R3 3383/4885
US-20240277694-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 KAT6A 3520/4885MGLL 2015/4885TAS1R3 3383/4885
US-20250243177-A1 sGC STIMULATORS GUCY1A1, PTGIS, GUCY1B1 KAT6A 3925/4885MGLL 2096/4885TAS1R3 1316/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.