SCHEMBL24869145

SCHEMBL24869145

CCCc1cnc(N)c(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
PKM P14618 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MAP3K12 Q12852 6/20 0.36
PIK3CA P42336 7/20 0.36
MTOR P42345 1/20 0.35
CYP3A4 P08684 1/20 0.35
PIK3CD O00329 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
PIK3C3 Q8NEB9 1/20 0.35
PI4KB Q9UBF8 1/20 0.35
DDR1 Q08345 1/20 0.35
NOS2 P35228 1/20 0.35
AR P10275 1/20 0.35
USP7 Q93009 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10268251 0.86 MTOR (0.40) MAP3K12PIK3CAMTORCYP3A4DDR1
SCHEMBL15412486 0.76 NOS2 (0.39) MAP3K12PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL11745802 0.76 NPC1 (0.44) NPC1TP53PKMRAB9ASMN1; SMN2
SCHEMBL11890838 0.72 NOS3 (0.54) HSD17B10MAP3K12PIK3CAMTORPIK3CD
SCHEMBL21503558 0.71 NPC1 (0.35) NPC1TP53PKMRAB9ASMN1; SMN2
SCHEMBL28844850 0.71 FFAR4 (0.47) NPC1TP53PKMRAB9ASMN1; SMN2
SCHEMBL21031807 0.71 GLA (0.45) MAP3K12PIK3CAMTORPIK3CDPIK3CB
SCHEMBL29601287 0.71 GLA (0.45) MAP3K12PIK3CAMTORPIK3CDPIK3CB
SCHEMBL20458857 0.71 MAP3K12 (0.39) NPC1RAB9AMAP3K12PIK3CAMTOR
SCHEMBL26563578 0.71 PARP1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023279986-A1 SIX-MEMBERED ARYL OR HETEROARYL AMIDES, AND COMPOSITION AND USE THEREOF 贝达药业股份有限公司 2023-01-12 WO disclosed