SCHEMBL24869253

SCHEMBL24869253

CC(C)c1cnc(N2C[C@H]3CC(=O)C[C@H]3C2)c(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.36
HRH3 Q9Y5N1 2/20 0.36
KCNH2 Q12809 1/20 0.36
P2RY12 Q9H244 2/20 0.34
ACACB O00763 3/20 0.33
PHGDH O43175 2/20 0.32
CXCR3 P49682 2/20 0.32
TRPV1 Q8NER1 2/20 0.32
KCNJ5 P48544 1/20 0.32
KCNJ3 P48549 1/20 0.32
HSD11B1 P28845 1/20 0.31
IDH1 O75874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16248222 0.75 P2RY12 (0.40) P2RY12TRPV1
SCHEMBL14349216 0.74 P2RY12 (0.39) P2RY12TRPV1
SCHEMBL24869248 0.72 P2RX7 (0.36) HRH4HRH3KCNH2P2RY12ACACB
SCHEMBL15599194 0.71 CHRNB2 (0.47) HRH4
SCHEMBL12891545 0.71 GRM4 (0.41) P2RY12
SCHEMBL21470275 0.71 LMNA (0.47)
SCHEMBL24869545 0.71 HRH4 (0.33) HRH4HRH3KCNH2P2RY12CXCR3
SCHEMBL21030633 0.68 MALT1 (0.44)
SCHEMBL24869254 0.68 GLP1R (0.46) P2RY12TRPV1
SCHEMBL17244900 0.68 P2RX7 (0.37) HRH4HRH3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023279986-A1 SIX-MEMBERED ARYL OR HETEROARYL AMIDES, AND COMPOSITION AND USE THEREOF 贝达药业股份有限公司 2023-01-12 WO disclosed