SCHEMBL2487771

SCHEMBL2487771

CCCCc1cc(N)cc(C(=O)O)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 8/20 0.51
CTRC Q99895 1/20 0.46
ALDH1A1 P00352 3/20 0.45
MEN1 O00255 2/20 0.45
MAPT P10636 2/20 0.45
KMT2A Q03164 2/20 0.45
RARA P10276 1/20 0.45
MTOR P42345 1/20 0.45
HPGD P15428 2/20 0.43
HSD17B10 Q99714 1/20 0.43
PLA2G2A P14555 1/20 0.42
GPR84 Q9NQS5 2/20 0.42
GABRP O00591 1/20 0.42
GABRD O14764 1/20 0.42
GABRA1 P14867 1/20 0.42
GABRB1 P18505 1/20 0.42
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA5 P31644 1/20 0.42
GABRA3 P34903 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28376268 0.89 TPMT (0.42) RARBALDH1A1MEN1MAPTKMT2A
SCHEMBL914005 0.87 RARB (0.59) RARBCTRCALDH1A1MEN1MAPT
SCHEMBL9701286 0.87 RARB (0.59) RARBCTRCALDH1A1MEN1MAPT
SCHEMBL27854912 0.85 GPR84 (0.41) RARBALDH1A1HPGDHSD17B10GPR84
SCHEMBL2725031 0.82 ALDH1A1 (0.50) ALDH1A1MEN1MAPTKMT2AHPGD
Octane SCHEMBL7266397 0.82 PLA2G2A (0.56) RARBALDH1A1MEN1MAPTKMT2A
SCHEMBL27782228 0.82 GPR84 (0.61) RARBALDH1A1MEN1MAPTKMT2A
SCHEMBL32679274 0.82 ALDH1A1 (0.50) ALDH1A1MEN1MAPTKMT2AHPGD
SCHEMBL8413501 0.82 RARB (0.61) RARBALDH1A1MEN1MAPTKMT2A
SCHEMBL25402608 0.81 PTGS2 (0.58) RARBCTRCALDH1A1MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379513-A1 HETEROARYL COMPOUNDS USEFUL AS RAF KINASE INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2011-10-26 EP disclosed
WO-2010078408-A1 HETEROARYL COMPOUNDS USEFUL AS RAF KINASE INHIBITORS BIOGEN IDEC MA INC. (US) 2010-07-08 WO disclosed