SCHEMBL2487994

SCHEMBL2487994

COC(=O)CC1CCC(F)(F)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.39
NR1H2 P55055 1/20 0.39
HSD17B10 Q99714 3/20 0.34
CYP3A4 P08684 1/20 0.34
MAPT P10636 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
APLNR P35414 1/20 0.33
SCN9A Q15858 5/20 0.32
TSHR P16473 3/20 0.32
GAA P10253 2/20 0.32
NAAA Q02083 1/20 0.32
ASAH1 Q13510 1/20 0.32
P2RX7 Q99572 2/20 0.31
EPHX2 P34913 1/20 0.31
PRKCA P17252 2/20 0.31
SCN5A Q14524 1/20 0.30
MGAM O43451 1/20 0.30
SI P14410 1/20 0.30
MGAM2 Q2M2H8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6344069 0.89 BRD4 (0.41) BRD4NR1H2HSD17B10CYP3A4MAPT
Hydrochloric Acid SCHEMBL28770722 0.87 BRD4 (0.40) BRD4NR1H2HSD17B10CYP3A4MAPT
SCHEMBL15106713 0.85 BRD4 (0.43) BRD4NR1H2HSD17B10CYP3A4MAPT
SCHEMBL20403281 0.83 NR1H2 (0.36) BRD4NR1H2EPHX2
SCHEMBL12206362 0.83 ALDH1A1 (0.38) HSD17B10APLNRTSHRGAAEPHX2
SCHEMBL51471 0.79 BRD4 (0.39) BRD4NR1H2HSD17B10TSHRGAA
SCHEMBL12561079 0.77 SCN9A (0.34) BRD4SCN9ATSHRGAANAAA
SCHEMBL29224201 0.77 SLC6A1 (0.39) MAPTAPLNR
SCHEMBL3185201 0.77 SLC6A1 (0.39) MAPTAPLNR
SCHEMBL29067928 0.76 BRD4 (0.37) BRD4NR1H2APLNRTSHRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102712577-B Substituted 3-phenylpropionic acids and the use thereof BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-10-15 CN disclosed
CN-103796989-A Branched 3-phenylpropionic acid derivatives and uses thereof BAYER IP GMBH 2014-05-14 CN disclosed
CN-103492361-A Substituted 1-benzylcycloalkylcarboxlic acids and use thereof BAYER IP GMBH 2014-01-01 CN disclosed
CN-102712577-A Substituted 3-phenylpropionic acids and the use thereof BAYER SCHERING PHARMA AG 2012-10-03 CN disclosed
EP-1697311-B1 NITRILE COMPOUND AND ITS USE IN PEST CONTROL SUMITOMO CHEMICAL CO (JP) 2011-10-26 EP disclosed
US-7662402-B2 contains fluoroalkyl group; insecticides, miticides, nematocides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2010-02-16 US disclosed
US-7662402-B2 contains fluoroalkyl group; insecticides, miticides, nematocides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2010-02-16 US disclosed
US-7662402-B2 contains fluoroalkyl group; insecticides, miticides, nematocides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2010-02-16 US disclosed
CN-100390140-C Nitrile compounds and their use in pest control SUMITOMO CHEMICAL CO (JP) 2008-05-28 CN disclosed
US-20070112068-A1 Nitrile compound and its use in pest control SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2007-05-17 US disclosed
US-20070112068-A1 Nitrile compound and its use in pest control SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2007-05-17 US disclosed
US-20070112068-A1 Nitrile compound and its use in pest control SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2007-05-17 US disclosed
CN-1898200-A Nitrile compound and its pest control use SUMITOMO CHEMICAL CO (JP) 2007-01-17 CN disclosed
EP-1697311-A1 NITRILE COMPOUND AND ITS USE IN PEST CONTROL Sumitomo Chemical Company, Limited (JP) 2006-09-06 EP disclosed
WO-2005063694-A1 NITRILE COMPOUND AND ITS USE IN PEST CONTROL SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2005-07-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070112068-A1 Nitrile compound and its use in pest control C5, C9, C1S BRD4 1585/4885NR1H2 2160/4885HSD17B10 2825/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.