SCHEMBL2488025

SCHEMBL2488025

CN(C)c1ccc(-c2ccc(Cn3cc(OC(=O)O)c(=O)c4c(F)ccc(F)c43)c(F)c2)cn1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 4/20 0.41
GRIN2B Q13224 11/20 0.35
GRIN1 Q05586 3/20 0.35
NPC1 O15118 1/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35
RAB9A P51151 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
GRM2 Q14416 1/20 0.33
ICMT O60725 1/20 0.32
KCNH2 Q12809 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2492205 0.89 CHRM1 (0.41) CHRM1GRIN2BGRIN1
SCHEMBL2491881 0.88 ERN1 (0.42) CHRM1GRIN2BGRIN1HDAC6
SCHEMBL2488465 0.88 CHRM1 (0.41) CHRM1GRIN2BGRIN1
SCHEMBL2488023 0.86 CHRM1 (0.54) CHRM1GRIN2BGRIN1NPC1POLB
SCHEMBL2492208 0.84 CHRM1 (0.41) CHRM1GRIN2BGRIN1
SCHEMBL2486084 0.84 CHRM1 (0.53) CHRM1RXFP1
SCHEMBL2487909 0.84 CHRM1 (0.43) CHRM1
SCHEMBL2488348 0.84 CHRM1 (0.40) CHRM1GRIN2B
SCHEMBL2487485 0.82 CHRM1 (0.45) CHRM1GRIN2BGRIN1
SCHEMBL2487494 0.80 CHRM1 (0.40) CHRM1ICMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2037739-B1 BENZYL-SUBSTITUTED QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK SHARP & DOHME (US) 2011-10-26 EP claimed