SCHEMBL2490903

SCHEMBL2490903

N#CSC(C=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACP3 P15309 3/20 0.41
CES2 O00748 2/20 0.41
PNMT P11086 1/20 0.41
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
DAO P14920 1/20 0.37
EPHX1 P07099 2/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
CTSS P25774 1/20 0.35
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
LRRK2 Q5S007 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2494300 0.81 KIF11 (0.37) ACP3CES2
SCHEMBL11156832 0.77 ACP3 (0.44) ACP3CES2PNMTIDO1TDO2
SCHEMBL23628841 0.76 TSHR (0.38) TSHRMAPK1
SCHEMBL4068170 0.76 TSHR (0.38) TSHRMAPK1
SCHEMBL15331089 0.74 ACP3 (0.50) ACP3CES2PNMTIDO1TDO2
SCHEMBL6970288 0.74 ACP3 (0.50) ACP3CES2PNMTIDO1TDO2
SCHEMBL5990120 0.71 CES2 (0.43) ACP3CES2PNMTIDO1TDO2
SCHEMBL17515119 0.71 DAO (0.49) ACP3CES2PNMTIDO1TDO2
SCHEMBL9570750 0.71 ACP3 (0.47) ACP3CES2PNMTIDO1TDO2
SCHEMBL1712441 0.71 PNMT (0.56) ACP3CES2PNMTIDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379543-A2 THIAZOLYL-BENZIMIDAZOLES F. Hoffmann-La Roche AG (CH) 2011-10-26 EP disclosed
WO-2010121675-A2 THIAZOLYL-BENZIMIDAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed