SCHEMBL24920567

SCHEMBL24920567

COCc1ccnc(N2CC3(CCOCC3)C2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.38
TTK P33981 1/20 0.37
PDCD1LG2 Q9BQ51 1/20 0.36
CD274 Q9NZQ7 1/20 0.36
HSD17B10 Q99714 5/20 0.36
ALDH1A1 P00352 5/20 0.36
HPGD P15428 4/20 0.36
CYP3A4 P08684 2/20 0.35
USP2 O75604 1/20 0.35
CYP2D6 P10635 2/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
AOC3 Q16853 1/20 0.35
CYP1A2 P05177 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
RXRA P19793 5/20 0.34
GRIN1 Q05586 5/20 0.34
GRIN2B Q13224 5/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24920538 0.91 DYRK1A (0.44) DYRK1AHSD17B10ALDH1A1CYP3A4USP2
SCHEMBL24920525 0.88 DYRK1A (0.52) DYRK1ATTKHSD17B10CYP3A4CYP2D6
SCHEMBL24920536 0.82 ACHE (0.48) ALDH1A1HPGDCYP3A4CYP2D6LMNA
SCHEMBL24920534 0.81 HSD17B10 (0.45) HSD17B10ALDH1A1HPGDCYP3A4USP2
SCHEMBL24921025 0.81 RXRA (0.39) DYRK1AAOC3RXRAGRIN1GRIN2B
SCHEMBL24921032 0.80 AOC3 (0.39) DYRK1AAOC3RXRAGRIN1GRIN2B
SCHEMBL24920516 0.80 HSD17B10 (0.41) DYRK1AHSD17B10ALDH1A1HPGDCYP3A4
SCHEMBL24920535 0.78 SLC6A2 (0.40) ALDH1A1HPGDHTTL3MBTL1AOC3
SCHEMBL24921023 0.76 AOC3 (0.44) DYRK1AAOC3RXRAGRIN1GRIN2B
SCHEMBL24921040 0.76 AOC3 (0.44) DYRK1AHTTAOC3RXRAGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed