SCHEMBL24920536

SCHEMBL24920536

COCc1ccnc(N2CCOCC2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.48
PIK3CA P42336 2/20 0.48
PIK3CD O00329 1/20 0.48
PIK3R1 P27986 1/20 0.48
PIK3CB P42338 1/20 0.48
MTOR P42345 5/20 0.46
MAPK1 P28482 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
ALDH1A1 P00352 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
EIF2AK2 P19525 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
GAA P10253 1/20 0.43
HPGD P15428 1/20 0.43
KMT2A Q03164 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24921023 0.88 AOC3 (0.44) ACHEKDM4EKMT2ACA12CA1
SCHEMBL24921040 0.88 AOC3 (0.44) ACHEMEN1KMT2ACA12CA1
SCHEMBL24920520 0.86 MAPT (0.46) ACHEMEN1HPGDKMT2ACA12
SCHEMBL24920548 0.85 ACHE (0.48) ACHEALDH1A1MEN1KMT2ACA12
SCHEMBL24920535 0.84 SLC6A2 (0.40) ACHEPIK3CAPIK3CDPIK3R1PIK3CB
SCHEMBL24920523 0.84 ADRB1 (0.51) ACHEALDH1A1KDM4EHPGDCYP1A2
SCHEMBL17827961 0.83 PIK3CA (0.51) ACHEPIK3CAPIK3CDPIK3R1PIK3CB
SCHEMBL24920567 0.82 DYRK1A (0.38) ACHEALDH1A1L3MBTL1HPGDCA12
SCHEMBL20745766 0.82 CA12 (0.47) ACHEPIK3CAPIK3CDPIK3R1PIK3CB
SCHEMBL24920538 0.82 DYRK1A (0.44) ALDH1A1L3MBTL1CYP3A4CYP2D6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed