SCHEMBL24920807

SCHEMBL24920807

COc1ncc(F)c(-c2nnc(C)o2)n1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 4/20 0.36
PTGDR Q13258 1/20 0.34
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.32
NOTUM Q6P988 1/20 0.32
BRD4 O60885 1/20 0.31
ATR Q13535 2/20 0.31
CYP1A2 P05177 2/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
AOC3 Q16853 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GLA P06280 1/20 0.30
CYP3A4 P08684 1/20 0.30
KMT2A Q03164 1/20 0.30
HIF1A Q16665 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24920864 0.76 MAPT (0.39) JAK1TYK2NOTUMNPC1RAB9A
SCHEMBL24920831 0.76 LRRK2 (0.36) LRRK2AOC3
SCHEMBL30822678 0.74 QPCT (0.40) LRRK2PTGDRNOTUMBRD4CYP1A2
SCHEMBL29164610 0.74 QPCT (0.40) LRRK2PTGDRNOTUMBRD4CYP1A2
SCHEMBL24920816 0.74 PDE10A (0.31) CYP1A2MEN1ALDH1A1GLACYP3A4
SCHEMBL24921547 0.74 NPC1 (0.37) LRRK2PTGDRJAK1TYK2BRD4
SCHEMBL24921525 0.74 NPC1 (0.40) PTGDRBRD4NPC1RAB9AAOC3
SCHEMBL24920782 0.73 PIM1 (0.36) LRRK2JAK1TYK2NOTUMBRD4
SCHEMBL24920776 0.73 L3MBTL1 (0.36) TRPM8NPC1RAB9AAOC3ALDH1A1
SCHEMBL24921979 0.71 PTGDR (0.39) LRRK2PTGDRNOTUMBRD4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed