SCHEMBL24920864

SCHEMBL24920864

COc1ncc(F)c(-c2nnco2)n1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.39
NOTUM Q6P988 10/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
MAPK1 P28482 1/20 0.38
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
GAA P10253 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
JAK1 P23458 1/20 0.32
TYK2 P29597 1/20 0.32
EDNRA P25101 1/20 0.31
TSHR P16473 1/20 0.31
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24920807 0.76 LRRK2 (0.36) NOTUMALDH1A1NPC1RAB9AJAK1
SCHEMBL24920816 0.74 PDE10A (0.31) ALDH1A1
SCHEMBL24921557 0.74 MAPT (0.53) MAPTNOTUMALDH1A1HPGDMAPK1
SCHEMBL24921606 0.73 NOTUM (0.47) MAPTNOTUMALDH1A1HPGDMAPK1
SCHEMBL24920831 0.73 LRRK2 (0.36) LMNA
SCHEMBL24920810 0.73 MAPT (0.39) MAPTNOTUMALDH1A1HPGDMAPK1
SCHEMBL24921973 0.71 MAPT (0.42) MAPTNOTUMALDH1A1HPGDMAPK1
SCHEMBL24920818 0.71 CYP1A2 (0.33) ALDH1A1HPGDMAPK1TSHR
SCHEMBL21905028 0.70 CYP1A2 (0.37) ALDH1A1MAPK1TSHR
SCHEMBL24920772 0.69 NOTUM (0.45) MAPTNOTUMALDH1A1HPGDMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed