SCHEMBL24920822

SCHEMBL24920822

COc1cc(-c2ncon2)ncn1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.48
CYP2C19 P33261 3/20 0.37
CNR2 P34972 1/20 0.35
CYP1A1 P04798 1/20 0.34
CYP1B1 Q16678 1/20 0.34
NPC1 O15118 2/20 0.30
RAB9A P51151 2/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MAPT P10636 1/20 0.30
NFKB1 P19838 1/20 0.30
NFKB2 Q00653 1/20 0.30
RELA Q04206 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24921178 0.75 BTK (0.42) KMO
SCHEMBL14447596 0.74 KMO (0.44) KMOCYP2C19CNR2NPC1RAB9A
SCHEMBL24921969 0.74 KMO (0.39) KMOCNR2NPC1RAB9AKDM4E
SCHEMBL24921988 0.74 CNR2 (0.36) KMOCNR2
SCHEMBL24920871 0.73 L3MBTL1 (0.41) CYP2C19NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL5347158 0.71 NPC1 (0.43) KMOCYP2C19NPC1RAB9ACYP1A2
SCHEMBL24921190 0.71 S1PR1 (0.49)
SCHEMBL24921180 0.71 CCR1 (0.61) KMOCYP2C19CNR2CYP1A1CYP1B1
SCHEMBL24920817 0.71 CYP11B2 (0.38) KMOCNR2
SCHEMBL14031855 0.70 CYP2C19 (0.41) CYP2C19CYP1A1CYP1B1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed