SCHEMBL24920818

SCHEMBL24920818

COc1ncc(F)c(-c2ncon2)n1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 5/20 0.33
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HDAC5 Q9UQL6 1/20 0.31
HSD17B10 Q99714 4/20 0.31
ALDH1A1 P00352 3/20 0.31
CYP3A4 P08684 3/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
GLA P06280 1/20 0.31
HIF1A Q16665 1/20 0.31
CYP2C9 P11712 2/20 0.30
TSHR P16473 1/20 0.30
MAPK1 P28482 1/20 0.30
USP2 O75604 1/20 0.30
CASP1 P29466 1/20 0.30
CASP7 P55210 1/20 0.30
HPGD P15428 1/20 0.30
CYP2C19 P33261 1/20 0.30
PPARA Q07869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24920776 0.77 L3MBTL1 (0.36) HDAC1HDAC6HDAC5HSD17B10ALDH1A1
SCHEMBL24920793 0.73 GUCY1B2 (0.40) KMT2APPARA
SCHEMBL24921552 0.73 FTO (0.37) PPARA
SCHEMBL24921572 0.72 PDK2 (0.34) HDAC1HDAC6HDAC5
SCHEMBL24920896 0.72 CYP1A2 (0.31) CYP1A2HSD17B10ALDH1A1CYP3A4MEN1
SCHEMBL24920831 0.71 LRRK2 (0.36) HDAC1HDAC6HDAC5
SCHEMBL24920864 0.71 MAPT (0.39) ALDH1A1TSHRMAPK1HPGD
SCHEMBL24921985 0.69 CNR2 (0.33)
SCHEMBL24920816 0.69 PDE10A (0.31) CYP1A2HSD17B10ALDH1A1CYP3A4MEN1
SCHEMBL21905028 0.68 CYP1A2 (0.37) CYP1A2HSD17B10ALDH1A1CYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed