SCHEMBL24921972

SCHEMBL24921972

COc1ccc(-c2ncno2)nn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.35
NNMT P40261 1/20 0.33
MAPT P10636 5/20 0.33
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
LMNA P02545 2/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
PPARG P37231 1/20 0.32
DUSP3 P51452 1/20 0.32
PTPN5 P54829 1/20 0.32
PTPN11 Q06124 1/20 0.32
NR2E3 Q9Y5X4 1/20 0.32
NCOR2 Q9Y618 1/20 0.32
SCD5 Q86SK9 2/20 0.32
SCD O00767 1/20 0.32
PDE10A Q9Y233 1/20 0.31
KDM4E B2RXH2 2/20 0.30
PKM P14618 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24921238 0.76 BTK (0.42) MAPTNPC1RAB9APDE10AKDM4E
SCHEMBL24920820 0.75 CYP2C19 (0.38) MAPTNPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL24921976 0.75 SIRT6 (0.36) PDE10A
SCHEMBL24921964 0.74 PDE10A (0.31) PDE10A
SCHEMBL24921577 0.74 CA1 (0.47) NNMTCA1CA2
SCHEMBL24922001 0.74
SCHEMBL24921573 0.74 PDE10A (0.45) NPC1RAB9ACA1CA2SCD5
SCHEMBL1456221 0.73 NNMT (0.46) MAOBNNMTMAPTNPC1RAB9A
SCHEMBL24920802 0.72 LRRK2 (0.38) PDE10A
SCHEMBL24921491 0.70 ACHE (0.42) MAOBMAPTNPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed