SCHEMBL24928843

SCHEMBL24928843

Cc1oncc1-c1cc(NS(=O)(=O)c2cc(C(=O)O)ccc2C2CC2)c(OC2CCC2)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACLY P53396 5/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
POLB P06746 1/20 0.36
HSD17B10 Q99714 1/20 0.36
RAD52 P43351 1/20 0.35
FABP4 P15090 1/20 0.35
PTGDR Q13258 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
PTK2B Q14289 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
NPC1 O15118 1/20 0.35
ERAP1 Q9NZ08 1/20 0.34
SCN5A Q14524 1/20 0.34
SCN9A Q15858 1/20 0.34
BRD4 O60885 1/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30153324 1.00 ACLY (0.38) ACLYL3MBTL1POLBHSD17B10RAD52
SCHEMBL24928651 0.98 ACLY (0.38) ACLYL3MBTL1POLBHSD17B10RAD52
SCHEMBL31198500 0.98 ACLY (0.38) ACLYL3MBTL1POLBHSD17B10RAD52
SCHEMBL30153260 0.94 ACLY (0.40) ACLYL3MBTL1PTGDRPTGDR2SMN1; SMN2
SCHEMBL30845553 0.94 ACLY (0.40) ACLYL3MBTL1PTGDRPTGDR2SMN1; SMN2
SCHEMBL24928850 0.91 ACLY (0.36) ACLYL3MBTL1POLBHSD17B10RAD52
SCHEMBL30153306 0.91 ACLY (0.36) ACLYL3MBTL1POLBHSD17B10RAD52
SCHEMBL24928655 0.89 ACLY (0.41) ACLYRAD52FABP4PTK2BSMN1; SMN2
SCHEMBL31198427 0.89 ACLY (0.41) ACLYRAD52FABP4PTK2BSMN1; SMN2
SCHEMBL24928647 0.85 BRD4 (0.44) ACLYPOLBRAD52TDP1ERAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117881657-A Phenyl-sulfamoyl-benzoic acid derivatives as ERAP1 modulators 格雷沃尔夫治疗有限公司 2024-04-12 CN disclosed
WO-2023007188-A1 PHENYL-SULFAMOYL-BENZOIC ACID DERIVATIVES AS ERAP1- MODULATORS Grey Wolf Therapeutics Limited (GB) 2023-02-02 WO disclosed