SCHEMBL24933186

SCHEMBL24933186

NC(=O)c1cc(-c2cccc(N)c2)c(C(F)(F)F)[nH]c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 8/20 0.44
HSD17B2 P37059 8/20 0.44
PARP1 P09874 3/20 0.43
PLK4 O00444 1/20 0.38
MAP4K4 O95819 1/20 0.38
EGFR P00533 1/20 0.38
ROS1 P08922 1/20 0.38
PIM1 P11309 1/20 0.38
AXL P30530 1/20 0.38
FLT3 P36888 1/20 0.38
FRK P42685 1/20 0.38
MAP4K2 Q12851 1/20 0.38
NTRK3 Q16288 1/20 0.38
MINK1 Q8N4C8 1/20 0.38
AURKB Q96GD4 1/20 0.38
HIPK2 Q9H2X6 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
STK17A Q9UEE5 1/20 0.38
ALK Q9UM73 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24932959 0.87 HSD17B1 (0.44) HSD17B1HSD17B2PARP1PDE3BPDE3A
SCHEMBL24932950 0.87 HSD17B2 (0.52) HSD17B1HSD17B2PARP1PDE3BPDE3A
SCHEMBL24933754 0.86 HSD17B2 (0.53) HSD17B1HSD17B2BRD4
SCHEMBL30896148 0.86 HSD17B2 (0.53) HSD17B1HSD17B2BRD4
SCHEMBL24933185 0.84 PARP1 (0.46) HSD17B1HSD17B2PARP1SCN9A
SCHEMBL24933348 0.83 CDC7 (0.47) HSD17B1HSD17B2PARP1
SCHEMBL24933175 0.81 HSD17B1 (0.42) HSD17B1HSD17B2PARP1SCN9A
SCHEMBL30240765 0.81 MAOB (0.47) PARP1
SCHEMBL24933605 0.80 HSD17B2 (0.41) HSD17B1HSD17B2PARP1PDE3BPDE3A
SCHEMBL24933312 0.80 BTK (0.42) HSD17B1HSD17B2PLK4MAP4K4ROS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240360082-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2024-10-31 US claimed
EP-4373809-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2024-05-29 EP claimed
CN-117980292-A Substituted pyridone compounds for the treatment of orthomyxoviral infections 诺华股份有限公司 2024-05-03 CN claimed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO claimed
US-20240360082-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2024-10-31 US disclosed
EP-4373809-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2024-05-29 EP disclosed
CN-117980292-A Substituted pyridone compounds for the treatment of orthomyxoviral infections 诺华股份有限公司 2024-05-03 CN disclosed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240360082-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS PNPO, PDXK, PLPBP HSD17B1 2274/4885HSD17B2 2882/4885PARP1 4171/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.