SCHEMBL24933333

SCHEMBL24933333

NC(=O)c1cc(-c2ccc(Oc3ccccc3)cc2)c(C(F)(F)F)[nH]c1=O

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GSTP1 P09211 1/20 0.44
CHEK2 O96017 4/20 0.44
HSD17B1 P14061 2/20 0.44
HSD17B2 P37059 2/20 0.44
PARP10 Q53GL7 1/20 0.41
BRD4 O60885 1/20 0.40
GPR84 Q9NQS5 1/20 0.40
CTNNB1 P35222 1/20 0.40
LCK P06239 1/20 0.39
SRC P12931 1/20 0.39
CSK P41240 1/20 0.39
BTK Q06187 3/20 0.39
XDH P47989 1/20 0.38
BACE1 P56817 1/20 0.38
SCN9A Q15858 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24932950 0.89 HSD17B2 (0.52) HSD17B1HSD17B2BRD4SCN9A
SCHEMBL24933349 0.85 GSTP1 (0.50) GSTP1CHEK2HSD17B1HSD17B2PARP10
SCHEMBL24933053 0.85 KDM4E (0.44) HSD17B1HSD17B2
SCHEMBL30896275 0.85 LMNA (0.45) HSD17B1HSD17B2
SCHEMBL24933007 0.84 PPARD (0.44) HSD17B1HSD17B2
SCHEMBL24933335 0.83 HSD17B2 (0.44) HSD17B1HSD17B2
SCHEMBL24933256 0.83 PDK2 (0.43) CHEK2HSD17B1HSD17B2BRD4XDH
SCHEMBL24933605 0.82 HSD17B2 (0.41) HSD17B1HSD17B2XDH
SCHEMBL24933312 0.82 BTK (0.42) CHEK2HSD17B1HSD17B2BTK
SCHEMBL24933359 0.81 HSD17B2 (0.50) HSD17B1HSD17B2BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240360082-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2024-10-31 US claimed
EP-4373809-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2024-05-29 EP claimed
CN-117980292-A Substituted pyridone compounds for the treatment of orthomyxoviral infections 诺华股份有限公司 2024-05-03 CN claimed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO claimed
US-20240360082-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2024-10-31 US disclosed
EP-4373809-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2024-05-29 EP disclosed
CN-117980292-A Substituted pyridone compounds for the treatment of orthomyxoviral infections 诺华股份有限公司 2024-05-03 CN disclosed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240360082-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS PNPO, PDXK, PLPBP GSTP1 3746/4885CHEK2 985/4885HSD17B1 2274/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.