SCHEMBL24933360

SCHEMBL24933360

CCc1cccc(NC(=O)c2cccnc2)c1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.73
SMN1; SMN2 Q16637 2/20 0.73
NPC1 O15118 2/20 0.73
KCNK3 O14649 1/20 0.68
TRPV1 Q8NER1 1/20 0.65
TSHR P16473 2/20 0.64
HTT P42858 1/20 0.64
LMNA P02545 1/20 0.64
HIF1A Q16665 1/20 0.64
MAPT P10636 3/20 0.64
NPSR1 Q6W5P4 2/20 0.64
USP2 O75604 1/20 0.64
TP53 P04637 1/20 0.64
MAPK1 P28482 1/20 0.64
KMT2A Q03164 3/20 0.63
CYP1A2 P05177 1/20 0.63
CYP2C9 P11712 1/20 0.63
MEN1 O00255 2/20 0.62
ALDH1A1 P00352 1/20 0.62
TDP1 Q9NUW8 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10076300 0.89 RAB9A (0.77) RAB9ASMN1; SMN2NPC1KCNK3TRPV1
SCHEMBL8252721 0.85 RAB9A (1.00) RAB9ASMN1; SMN2NPC1TRPV1LMNA
SCHEMBL22983352 0.83 ALDH1A1 (0.84) RAB9ASMN1; SMN2NPC1KCNK3TSHR
SCHEMBL12314962 0.83 KCNK9 (0.69) RAB9ASMN1; SMN2NPC1KCNK3HTT
SCHEMBL9979193 0.82 ALDH1A1 (0.62) RAB9ASMN1; SMN2NPC1KCNK3LMNA
SCHEMBL259177 0.82 TDP1 (0.78) RAB9ASMN1; SMN2NPC1KCNK3TSHR
SCHEMBL3637836 0.82 HDAC3 (0.65) RAB9ASMN1; SMN2NPC1KCNK3TSHR
SCHEMBL882779 0.82 KCNK3 (0.69) RAB9ASMN1; SMN2NPC1KCNK3TSHR
SCHEMBL13766306 0.81 SMN1; SMN2 (0.58) SMN1; SMN2TRPV1TSHRHTTLMNA
SCHEMBL8376717 0.81 NPC1 (0.72) RAB9ASMN1; SMN2NPC1TRPV1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023009475-A1 ROCK2 INHIBITORS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2023-02-02 WO disclosed