SCHEMBL2495065

SCHEMBL2495065

CN(C)C(=O)[C@@H]1C[C@@H](OCCO[Si](C)(C)C(C)(C)C)CN1C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
UCHL1 P09936 1/20 0.40
NR1H2 P55055 1/20 0.31
MCL1 Q07820 2/20 0.31
BCL2 P10415 1/20 0.30
BCL2L1 Q07817 1/20 0.30
P2RX3 P56373 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2496930 0.94 UCHL1 (0.39) UCHL1NR1H2MCL1BCL2BCL2L1
SCHEMBL5068395 0.88 UCHL1 (0.30) UCHL1
SCHEMBL2501733 0.84 UCHL1 (0.41) UCHL1NR1H2MCL1P2RX3
SCHEMBL2495165 0.82 UCHL1 (0.40) UCHL1NR1H2MCL1P2RX3
SCHEMBL5071356 0.81 AGTR2 (0.33)
SCHEMBL5352509 0.81 UCHL1 (0.42) UCHL1NR1H2MCL1P2RX3
SCHEMBL2499313 0.80 UCHL1 (0.39) UCHL1NR1H2MCL1
SCHEMBL2502694 0.77 UCHL1 (0.40) UCHL1NR1H2MCL1P2RX3
SCHEMBL2494481 0.77 UCHL1 (0.40) UCHL1NR1H2MCL1
SCHEMBL5359255 0.77 UCHL1 (0.54) UCHL1NR1H2MCL1P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8030499-B2 1,3-dihydro-2H-indole-2-one compound and pyrrolidine-2-one compound fused with aromatic heterocycle TAISHO PHARMACEUTICAL CO., LTD. (JP) 2011-10-04 US disclosed