SCHEMBL24959800

SCHEMBL24959800

CC(=O)c1ccc(CC(C)(C)F)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 6/20 0.42
NR1H4 Q96RI1 5/20 0.42
PKM P14618 1/20 0.40
ESRRA P11474 1/20 0.40
PDK1 Q15118 5/20 0.40
PDK2 Q15119 5/20 0.40
PDK3 Q15120 5/20 0.40
PDK4 Q16654 5/20 0.40
HTT P42858 2/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ADRB2 P07550 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.37
GGPS1 O95749 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16728864 0.79 TAS1R3 (0.49) EPHX2NR1H4PKMHTTMEN1
SCHEMBL30665778 0.77 CYP2D6 (0.42) EPHX2NR1H4PKMESRRAHTT
SCHEMBL17831661 0.77 CYP2D6 (0.42) EPHX2NR1H4PKMESRRAHTT
SCHEMBL16899217 0.77 EPHX2 (0.55) EPHX2NR1H4HTTMEN1LMNA
SCHEMBL15492066 0.76 PKM (0.44) EPHX2NR1H4PKMHTTMEN1
SCHEMBL4814551 0.75 PKM (0.43) EPHX2NR1H4PKMHTTMEN1
SCHEMBL4810977 0.75 PKM (0.47) EPHX2NR1H4PKMHTTMEN1
SCHEMBL4090026 0.73 HPGD (0.44) PKMHTTMEN1LMNAMAPT
SCHEMBL313146 0.73 KIF11 (0.54) ESRRAPDK1MRGPRX4MAOAMAOB
SCHEMBL15352043 0.71 MRGPRX4 (0.52) ESRRAHTTMEN1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023288253-A1 SMALL MOLECULES INHIBITORS OF CYCLIC GMP-AMP SYNTHASE (CGAS) THE SCRIPPS RESEARCH INSTITUTE (US) 2023-01-19 WO disclosed