SCHEMBL24959842

SCHEMBL24959842

O=C(Cl)c1ccc(COC(F)(F)F)c(F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.40
IDO1 P14902 3/20 0.36
EPHX2 P34913 1/20 0.35
NR1H4 Q96RI1 1/20 0.35
HDAC6 Q9UBN7 3/20 0.34
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
AGXT P21549 2/20 0.34
S1PR1 P21453 1/20 0.34
S1PR3 Q99500 1/20 0.34
ALDH1A1 P00352 1/20 0.33
ENPP2 Q13822 1/20 0.33
ATXN2 Q99700 1/20 0.33
CHRNA7 P36544 1/20 0.33
PARP15 Q460N3 1/20 0.33
PARP14 Q460N5 1/20 0.33
PARP10 Q53GL7 1/20 0.33
HDAC4 P56524 2/20 0.33
HDAC7 Q8WUI4 2/20 0.33
HDAC11 Q96DB2 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3049461 0.76 CES2 (0.41) MAOBEPHX2NR1H4HDAC6CES2
SCHEMBL4123049 0.76 CES2 (0.41) MAOBEPHX2NR1H4CES2CES1
SCHEMBL24956830 0.73 MRGPRX4 (0.55) EPHX2NR1H4ALDH1A1
SCHEMBL24956819 0.72 EPHX2 (0.55) EPHX2CES2CES1
SCHEMBL20115903 0.71 KIF11 (0.53) IDO1
SCHEMBL18707178 0.70 KDM4E (0.53) CES2CES1
SCHEMBL29470947 0.69 CES2 (0.67) CES2CES1ALDH1A1
SCHEMBL192962 0.69 CES2 (0.67) CES2CES1ALDH1A1
SCHEMBL30308280 0.69 KIF11 (0.56) CES2CES1
SCHEMBL662965 0.69 KIF11 (0.56) CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023288253-A1 SMALL MOLECULES INHIBITORS OF CYCLIC GMP-AMP SYNTHASE (CGAS) THE SCRIPPS RESEARCH INSTITUTE (US) 2023-01-19 WO disclosed