SCHEMBL2497084

SCHEMBL2497084

C[C@H](O[Si](C)(C)C(C)(C)C)c1ccc(B2OC(C)(C)C(C)(C)O2)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 3/20 0.41
EGFR P00533 2/20 0.36
LPL P06858 7/20 0.34
LIPG Q9Y5X9 7/20 0.34
SNCA P37840 1/20 0.33
DGAT1 O75907 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
PRMT5 O14744 1/20 0.32
WDR77 Q9BQA1 1/20 0.32
HIF1A Q16665 1/20 0.31
FFAR1 O14842 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14758481 0.82 AAK1 (0.40) AAK1EGFRLPLLIPGSNCA
SCHEMBL24252905 0.81 AAK1 (0.41) AAK1EGFRLPLLIPGDGAT1
SCHEMBL4578027 0.80 AAK1 (0.39) AAK1EGFRLPLLIPGSNCA
SCHEMBL9910113 0.76 PDE2A (0.44) AAK1EGFRLPLLIPGCA1
SCHEMBL3025664 0.76 LMNA (0.50) AAK1EGFRLPLLIPGCA1
SCHEMBL2699826 0.76 PDE2A (0.44) AAK1EGFRLPLLIPGCA1
SCHEMBL2411421 0.75 LPL (0.44) AAK1EGFRLPLLIPGCA1
SCHEMBL2500684 0.74 ESR1 (0.46)
SCHEMBL2497862 0.74 APLNR (0.46) AAK1
SCHEMBL25314604 0.73 AAK1 (0.39) AAK1LPLLIPGDGAT1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8030327-B2 3-[1-(2-chlorophenyl)ethoxy]-5-imidazo[1,2-a]pyridin-3-ylthiophene-2-carboxyamide; polo like kinase inhibitor; antitumor and anticarcinogenic agent; mitotic phase (M phase) of the cell cycle MDS K.K. (JP) 2011-10-04 US disclosed