SCHEMBL2497148

SCHEMBL2497148

Cc1c(-c2c[nH]nc2C2CCN(C)CC2)cnc(N)c1C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 3/20 0.34
HTR1A P08908 3/20 0.34
HTR1D P28221 3/20 0.34
HTR1F P30939 3/20 0.34
HTR1B P28222 2/20 0.34
PRKAB2 O43741 1/20 0.33
PRKAG1 P54619 1/20 0.33
PRKAA2 P54646 1/20 0.33
PRKAA1 Q13131 1/20 0.33
PRKAG3 Q9UGI9 1/20 0.33
PRKAG2 Q9UGJ0 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33
LRRK2 Q5S007 2/20 0.33
PIK3C3 Q8NEB9 1/20 0.32
PARP1 P09874 1/20 0.31
CDK1 P06493 1/20 0.31
STAT6 P42226 1/20 0.30
MAP3K12 Q12852 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3469349 0.79 BMPR1B (0.39) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL3952939 0.79 ATR (0.40) ATRHTR1AHTR1DHTR1FHTR1B
Hydrochloric Acid SCHEMBL3469292 0.78 BMPR1B (0.38) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL3469290 0.74 BMPR1B (0.38) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL3950236 0.74 ATR (0.40) ATRHTR1AHTR1DHTR1FHTR1B
SCHEMBL2497147 0.73 BMPR1B (0.40) LRRK2PIK3C3MAP4K1
SCHEMBL1559096 0.68 HTR1D (0.44) HTR1AHTR1DHTR1FHTR1B
SCHEMBL3469125 0.67 CHRNA7 (0.43)
SCHEMBL29136767 0.66 KDM4E (0.39) ATRPIK3C3KMT2A
SCHEMBL23012343 0.65 QDPR (0.44) HTR1AHTR1DHTR1FHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2215085-B1 PYRIDINE AND PYRAZINE DERIVATIVES USEFUL IN THE TREATMENT OF CELL PROLIFERATIVE DISORDERS ASTRAZENECA AB (SE) 2011-09-07 EP disclosed