SCHEMBL24975799

SCHEMBL24975799

CC(C)(C)OC(=O)N(Cc1ccc2nc(C=O)cc(-c3cccc4cccnc34)c2c1)C1CCOCC1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
REN P00797 1/20 0.33
CYP3A4 P08684 1/20 0.33
KCNH2 Q12809 1/20 0.33
NR1H4 Q96RI1 1/20 0.32
UBE2M P61081 1/20 0.32
DCUN1D1 Q96GG9 1/20 0.32
KDM4E B2RXH2 2/20 0.32
POLB P06746 1/20 0.32
HSD11B1 P28845 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PIK3C2B O00750 1/20 0.31
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30
GRM2 Q14416 1/20 0.30
SLC22A12 Q96S37 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31428796 1.00 REN (0.33) RENCYP3A4KCNH2NR1H4UBE2M
SCHEMBL31428883 0.90 MMP9 (0.36) RENCYP3A4KCNH2NR1H4UBE2M
SCHEMBL31428558 0.87 GRM2 (0.35) KCNH2NR1H4HSD11B1SLC6A2SLC6A4
SCHEMBL24975810 0.87 GRM2 (0.35) KCNH2NR1H4HSD11B1SLC6A2SLC6A4
SCHEMBL31428765 0.86 ALDH1A1 (0.32) NR1H4UBE2MDCUN1D1
SCHEMBL24975804 0.85 GRM2 (0.35) CYP3A4NR1H4HSD11B1SLC6A2SLC6A4
SCHEMBL31428746 0.85 GRM2 (0.35) CYP3A4NR1H4HSD11B1SLC6A2SLC6A4
SCHEMBL31428465 0.85 GRM2 (0.39) KCNH2NR1H4HSD11B1SLC6A2SLC6A4
SCHEMBL24975808 0.84 SLC6A2 (0.39) KCNH2NR1H4HSD11B1SLC6A2SLC6A4
SCHEMBL31428539 0.82 GRM2 (0.35) NR1H4GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023008577-A1 RAS/RAF BINDING INHIBITOR COMPOUND 国立大学法人神戸大学 2023-02-02 WO disclosed