SCHEMBL24976359

SCHEMBL24976359

COC(=O)c1ccc2c(cnn2-c2nccc(C)n2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.47
CYP11B2 P19099 2/20 0.47
ALOX15 P16050 2/20 0.43
HTT P42858 1/20 0.43
KDM4E B2RXH2 4/20 0.42
JMJD6 Q6NYC1 1/20 0.41
IRAK4 Q9NWZ3 2/20 0.41
SMO Q99835 1/20 0.41
MAPK1 P28482 4/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39
RAB9A P51151 1/20 0.39
KLF5 Q13887 1/20 0.39
CYP19A1 P11511 1/20 0.39
KDM6B O15054 1/20 0.39
KDM5C P41229 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21725159 0.86 IRAK4 (0.43) HTTKDM4EJMJD6IRAK4SMO
SCHEMBL348090 0.78 CYP11B1 (0.57) CYP11B1CYP11B2KDM4ESMORAB9A
SCHEMBL23535745 0.78 CYP11B1 (0.60) CYP11B1CYP11B2ALOX15HTTKDM4E
SCHEMBL30204271 0.77 ALOX15 (0.50) CYP11B1CYP11B2ALOX15HTTKDM4E
SCHEMBL20373135 0.76 CYP11B1 (0.47) CYP11B1CYP11B2ALOX15HTTKDM4E
SCHEMBL10559859 0.75 KMT2A (0.46) ALOX15KDM4ETSHRRAB9AKMT2A
SCHEMBL10515588 0.74 KMT2A (0.55) KDM4ELMNACYP1A2CYP2C9TSHR
SCHEMBL1363389 0.74 CYP11B1 (0.69) CYP11B1CYP11B2SMO
SCHEMBL10516201 0.74 KMT2A (0.45) ALOX15KDM4ETSHRRAB9AKMT2A
SCHEMBL1144917 0.74 PDE1C (0.57) CYP11B1CYP11B2ALOX15HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11572374-B2 N-cyano-7-azanorbornane derivatives and uses thereof AMGEN INC. (US) 2023-02-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11572374-B2 N-cyano-7-azanorbornane derivatives and uses thereof CYP3A7, CYP51A1, NT5C3B CYP11B1 83/4885CYP11B2 103/4885ALOX15 1742/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.