SCHEMBL25017484

SCHEMBL25017484

CON(C)C(=O)[C@H]1[C@@H]2CNC[C@@H]21

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 4/20 0.33
CHRNA4 P43681 4/20 0.33
CHRNB4 P30926 2/20 0.33
CHRNA3 P32297 2/20 0.33
SSTR4 P31391 2/20 0.33
CHRNA7 P36544 1/20 0.33
SRD5A2 P31213 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25699204 1.00 CHRNB2 (0.33) CHRNB2CHRNA4CHRNB4CHRNA3SSTR4
SCHEMBL25177787 1.00 CHRNB2 (0.33) CHRNB2CHRNA4CHRNB4CHRNA3SSTR4
SCHEMBL25699206 1.00 CHRNB2 (0.33) CHRNB2CHRNA4CHRNB4CHRNA3SSTR4
SCHEMBL25181707 0.88 SRD5A2 (0.31) SRD5A2
SCHEMBL23230398 0.81 CHRNB2 (0.43) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL7897282 0.79 CHRNB2 (0.39) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL14606051 0.79 SSTR4 (0.37) CHRNB2CHRNA4CHRNB4CHRNA3SSTR4
SCHEMBL29152674 0.79 SSTR4 (0.37) CHRNB2CHRNA4CHRNB4CHRNA3SSTR4
Hydrochloric Acid SCHEMBL21640846 0.78 CHRNB2 (0.38) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL21253155 0.78 ALOX15 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250340548-A1 KRAS G12C INHIBITORS FRONTIER MEDICINES CORP (US) 2025-11-06 US disclosed
US-12291539-B2 KRAS G12C inhibitors FRONTIER MEDICINES CORPORATION (US) 2025-05-06 US disclosed
US-20250019387-A1 KRAS G12C INHIBITORS FRONTIER MEDICINES CORPORATION 2025-01-16 US disclosed
EP-4426695-A1 KRAS G12C INHIBITORS Frontier Medicines Corporation (US) 2024-09-11 EP disclosed
WO-2023081840-A1 KRAS G12C INHIBITORS FRONTIER MEDICINES CORPORATION (US) 2023-05-11 WO disclosed
WO-2023081840-A1 KRAS G12C INHIBITORS FRONTIER MEDICINES CORPORATION (US) 2023-05-11 WO disclosed
US-20230023559-A1 ARYLMETHYLENE HETEROCYCLIC COMPOUNDS AS KV1.3 POTASSIUM SHAKER CHANNEL BLOCKERS D. E. SHAW RESEARCH, LLC (US) 2023-01-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12291539-B2 KRAS G12C inhibitors KRAS, NRAS, HRAS CHRNB2 4812/4885CHRNA4 4876/4885CHRNB4 4835/4885
US-20250340548-A1 KRAS G12C INHIBITORS KRAS, NRAS, HRAS CHRNB2 4812/4885CHRNA4 4876/4885CHRNB4 4835/4885
US-20230023559-A1 ARYLMETHYLENE HETEROCYCLIC COMPOUNDS AS KV1.3 POTASSIUM SHAKER CHANNEL BLOCKERS KCNJ2, KCNA3, KCNH3 CHRNB2 228/4885CHRNA4 259/4885CHRNB4 266/4885
US-20250019387-A1 KRAS G12C INHIBITORS KRAS, NRAS, HRAS CHRNB2 4812/4885CHRNA4 4876/4885CHRNB4 4835/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.