SCHEMBL25181707

SCHEMBL25181707

CON(C)C(=O)C1C2CCNCC21

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 1/20 0.31
SLC6A1 P30531 2/20 0.30
GABRA5 P31644 2/20 0.30
GABRB2 P47870 2/20 0.30
SLC6A12 P48065 2/20 0.30
SLC6A11 P48066 2/20 0.30
SLC6A13 Q9NSD5 2/20 0.30
GABRA1 P14867 1/20 0.30
GABRR1 P24046 1/20 0.30
GABRA4 P48169 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25699206 0.88 CHRNB2 (0.33) SRD5A2
SCHEMBL25017484 0.88 CHRNB2 (0.33) SRD5A2
SCHEMBL25699204 0.88 CHRNB2 (0.33) SRD5A2
SCHEMBL25177787 0.88 CHRNB2 (0.33) SRD5A2
SCHEMBL21253155 0.78 ALOX15 (0.35)
SCHEMBL25015548 0.77 REN (0.38) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
SCHEMBL20015534 0.77 REN (0.38) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
SCHEMBL13153259 0.77 REN (0.38) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
Hydrochloric Acid SCHEMBL25232390 0.76 REN (0.37) SLC6A1GABRA5GABRB2SLC6A12SLC6A11
Hydrochloric Acid SCHEMBL28945920 0.76 REN (0.37) SLC6A1GABRA5GABRB2SLC6A12SLC6A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250340548-A1 KRAS G12C INHIBITORS FRONTIER MEDICINES CORP (US) 2025-11-06 US disclosed
US-12291539-B2 KRAS G12C inhibitors FRONTIER MEDICINES CORPORATION (US) 2025-05-06 US disclosed
US-20250019387-A1 KRAS G12C INHIBITORS FRONTIER MEDICINES CORPORATION 2025-01-16 US disclosed
EP-4426695-A1 KRAS G12C INHIBITORS Frontier Medicines Corporation (US) 2024-09-11 EP disclosed
WO-2023081840-A1 KRAS G12C INHIBITORS FRONTIER MEDICINES CORPORATION (US) 2023-05-11 WO disclosed
WO-2023081840-A1 KRAS G12C INHIBITORS FRONTIER MEDICINES CORPORATION (US) 2023-05-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12291539-B2 KRAS G12C inhibitors KRAS, NRAS, HRAS SRD5A2 4522/4885SLC6A1 4613/4885GABRA5 4175/4885
US-20250340548-A1 KRAS G12C INHIBITORS KRAS, NRAS, HRAS SRD5A2 4522/4885SLC6A1 4613/4885GABRA5 4175/4885
US-20250019387-A1 KRAS G12C INHIBITORS KRAS, NRAS, HRAS SRD5A2 4522/4885SLC6A1 4613/4885GABRA5 4175/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.