SCHEMBL25041248

SCHEMBL25041248

O=c1[nH]c2ccc(/C=N/O)cc2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
PTK6 Q13882 7/20 0.41
GAA P10253 2/20 0.41
PKM P14618 1/20 0.41
MAPT P10636 2/20 0.40
KMT2A Q03164 1/20 0.40
PDE3B Q13370 2/20 0.40
PDE3A Q14432 2/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
GRIA1 P42261 3/20 0.38
CACNG8 Q8WXS5 2/20 0.38
GRIK1 P39086 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30275144 1.00 KDM4E (0.43) KDM4EALDH1A1L3MBTL1PTK6GAA
SCHEMBL30275170 1.00 KDM4E (0.43) KDM4EALDH1A1L3MBTL1PTK6GAA
Cyanide SCHEMBL22130260 0.77 GAA (0.41) KDM4EALDH1A1PTK6GAAPKM
SCHEMBL29519732 0.76 KIF11 (0.48) KDM4EALDH1A1GAAPKMMAPT
SCHEMBL1418732 0.76 KIF11 (0.48) KDM4EALDH1A1GAAPKMMAPT
SCHEMBL20493605 0.75 GAA (0.44) KDM4EALDH1A1GAAPKMMAPT
SCHEMBL20564646 0.73 NOS1 (0.51) KDM4EALDH1A1L3MBTL1GAAMAPT
SCHEMBL26977516 0.70 LMNA (0.47) KDM4EALDH1A1L3MBTL1GAAPKM
SCHEMBL12417111 0.70 MAPT (0.56) KDM4EALDH1A1PTK6MAPTKMT2A
SCHEMBL10139187 0.68 PTK6 (0.49) KDM4EALDH1A1PTK6GAAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115703768-A Compounds useful as inhibitors of ATR kinase 苏州爱科百发生物医药技术有限公司 2023-02-17 CN disclosed
WO-2023016525-A1 COMPOUND AS ATR KINASE INHIBITOR 苏州爱科百发生物医药技术有限公司 2023-02-16 WO disclosed