SCHEMBL25044720

SCHEMBL25044720

O=C(O)c1nnn(-c2ccc(C(F)F)cc2)c1COc1ccc(Cl)nn1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.36
GABRA5 P31644 6/20 0.35
GABRG2 P18507 4/20 0.35
GABRB3 P28472 4/20 0.35
KCNH2 Q12809 1/20 0.35
PTGS2 P35354 3/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA9 Q16790 1/20 0.33
RXRA P19793 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
TP53 P04637 1/20 0.32
ALOX12 P18054 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PPARG P37231 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30283031 1.00 HTT (0.36) HTTGABRA5GABRG2GABRB3KCNH2
SCHEMBL30282968 0.91 GABRA5 (0.36) GABRA5GABRG2GABRB3KCNH2PTGS2
SCHEMBL25044731 0.91 GABRA5 (0.36) GABRA5GABRG2GABRB3KCNH2PTGS2
SCHEMBL30282919 0.89 L3MBTL1 (0.45) GABRA5GABRG2GABRB3KCNH2PTGS2
SCHEMBL25044716 0.89 L3MBTL1 (0.45) GABRA5GABRG2GABRB3KCNH2PTGS2
SCHEMBL25045392 0.85 RXRA (0.33) GABRA5GABRG2GABRB3KCNH2RXRA
SCHEMBL30283165 0.85 RXRA (0.33) GABRA5GABRG2GABRB3KCNH2RXRA
SCHEMBL25045285 0.84 RXRA (0.33) GABRA5GABRG2GABRB3KCNH2RXRA
SCHEMBL27242697 0.83 ALDH1A1 (0.40) GABRA5GABRG2GABRB3KCNH2CA1
SCHEMBL21623964 0.83 GABRA5 (0.43) GABRA5GABRG2GABRB3KCNH2RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115703765-A Substituted triazole derivative, preparation method, pharmaceutical composition and application thereof 上海赛默罗生物科技有限公司 2023-02-17 CN disclosed
WO-2023016521-A1 SUBSTITUTED TRIAZOLE DERIVATIVE, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF 上海赛默罗生物科技有限公司 2023-02-16 WO disclosed