SCHEMBL25045281

SCHEMBL25045281

Fc1ccc(-n2nnc(Cl)c2COc2ccc(Cl)nn2)cc1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 12/20 0.41
GABRG2 P18507 9/20 0.41
GABRB3 P28472 9/20 0.41
KCNH2 Q12809 5/20 0.41
RXRA P19793 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25045411 0.90 NOTUM (0.37) GABRA5GABRG2GABRB3KCNH2RXRA
SCHEMBL2688352 0.88 GABRA5 (0.54) GABRA5GABRG2GABRB3KCNH2ALDH1A1
SCHEMBL30282901 0.88 GABRA5 (0.54) GABRA5GABRG2GABRB3KCNH2ALDH1A1
SCHEMBL30283165 0.86 RXRA (0.33) GABRA5GABRG2GABRB3KCNH2RXRA
SCHEMBL25045392 0.86 RXRA (0.33) GABRA5GABRG2GABRB3KCNH2RXRA
SCHEMBL27242729 0.85 GABRA5 (0.41) GABRA5GABRG2GABRB3KCNH2RXRA
SCHEMBL30282997 0.85 GABRA5 (0.41) GABRA5GABRG2GABRB3KCNH2RXRA
SCHEMBL30237297 0.80 BPTF (0.42) GABRA5GABRG2GABRB3KCNH2
SCHEMBL29036226 0.79 GABRG2 (0.38) GABRA5GABRG2GABRB3KCNH2RXRA
SCHEMBL25044752 0.77 GABRA5 (0.44) GABRA5GABRG2GABRB3KCNH2RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115703765-B Substituted triazole derivative, preparation method, pharmaceutical composition and application thereof 上海赛默罗生物科技有限公司 2025-02-28 CN disclosed
CN-115703765-A Substituted triazole derivative, preparation method, pharmaceutical composition and application thereof 上海赛默罗生物科技有限公司 2023-02-17 CN disclosed
WO-2023016521-A1 SUBSTITUTED TRIAZOLE DERIVATIVE, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF 上海赛默罗生物科技有限公司 2023-02-16 WO disclosed