SCHEMBL25087486

SCHEMBL25087486

COc1c(Br)cc(F)cc1[C@H](C)CO

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.38
CA2 P00918 2/20 0.35
CA4 P22748 2/20 0.35
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
ABCB11 O95342 1/20 0.34
NCOA1 Q15788 1/20 0.33
NCOA3 Q9Y6Q9 1/20 0.33
APLNR P35414 1/20 0.33
HSD17B10 Q99714 2/20 0.33
MAPK1 P28482 1/20 0.33
LMNA P02545 1/20 0.32
TPMT P51580 1/20 0.32
ALOX15 P16050 1/20 0.32
ALOX12 P18054 1/20 0.32
TSHR P16473 1/20 0.31
APOBEC3A P31941 1/20 0.31
HTT P42858 1/20 0.31
APOBEC3G Q9HC16 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31075666 0.74 ADRB2 (0.41) CA2CA4ABCB11HSD17B10TPMT
SCHEMBL31076037 0.74 ADRB2 (0.41) CA2CA4ABCB11HSD17B10TPMT
SCHEMBL31075853 0.74 ADRB2 (0.41) CA2CA4ABCB11HSD17B10TPMT
SCHEMBL1163205 0.74 CA2 (0.52) HTR2ACA2CA4MEN1MAPT
SCHEMBL31383825 0.73 APLNR (0.40) KMT2AAPLNR
SCHEMBL8165954 0.71 HTR2A (0.37) HTR2A
SCHEMBL8168673 0.71 HTR2A (0.37) HTR2A
SCHEMBL16737884 0.70 HTR2A (0.40) HTR2AABCB11HTT
SCHEMBL21787511 0.70 TRPA1 (0.33) HTR2AALOX15ALOX12
SCHEMBL21777352 0.70 TRPA1 (0.33) HTR2AALOX15ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023027948-A1 JAK2 INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2023-03-02 WO disclosed