SCHEMBL25113752

SCHEMBL25113752

COc1ccc(CN2C(=O)C(C)=C(Br)N(C)C2O)cc1OC

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
HTT P42858 3/20 0.43
MAPK10 P53779 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
KMT2A Q03164 2/20 0.41
HSP90AA1 P07900 1/20 0.40
LDHA P00338 1/20 0.40
MEN1 O00255 1/20 0.40
SMN1; SMN2 Q16637 5/20 0.40
LMNA P02545 5/20 0.40
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25113754 0.79 HSP90AA1 (0.39) ALDH1A1HTTSIGMAR1KMT2AHSP90AA1
SCHEMBL30323146 0.72 SIGMAR1 (0.48) ALDH1A1HTTSIGMAR1KMT2AHSP90AA1
SCHEMBL6552371 0.72 SIGMAR1 (0.48) ALDH1A1HTTSIGMAR1KMT2AHSP90AA1
SCHEMBL4628903 0.70 KMT2A (0.55) ALDH1A1HTTMAPK10SIGMAR1KMT2A
SCHEMBL27721661 0.65 LMNA (0.53) ALDH1A1HTTSIGMAR1KMT2AMEN1
SCHEMBL3470063 0.65 RGS4 (0.55) ALDH1A1HTTMAPK10SIGMAR1KMT2A
SCHEMBL15666947 0.64 MAPK10 (0.47) ALDH1A1HTTMAPK10SIGMAR1KMT2A
SCHEMBL12359560 0.64 KMT2A (0.50) ALDH1A1SIGMAR1KMT2AHSP90AA1MEN1
SCHEMBL2921022 0.64 SIGMAR1 (0.58) SIGMAR1KMT2AMEN1LMNA
SCHEMBL8242388 0.63 KMT2A (0.52) ALDH1A1KMT2ASMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3421462-B1 HETEROAROMATIC COMPOUNDS AND THEIR USE AS DOPAMINE D1 LIGANDS PFIZER (US) 2023-04-05 EP disclosed