SCHEMBL25193000

SCHEMBL25193000

COc1nc(-c2ccc(C(F)(F)F)nc2)ncc1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.41
TRPV3 Q8NET8 3/20 0.41
AURKA O14965 1/20 0.40
KDR P35968 1/20 0.40
AURKB Q96GD4 1/20 0.40
KMT2A Q03164 1/20 0.40
CASP3 P42574 1/20 0.38
TRPV4 Q9HBA0 1/20 0.38
KDM4E B2RXH2 1/20 0.37
PKM P14618 1/20 0.37
CHEK1 O14757 1/20 0.37
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
PI4KA P42356 1/20 0.36
PIK3CG P48736 1/20 0.36
PI4KB Q9UBF8 1/20 0.36
KCNH2 Q12809 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29635376 0.78 PDE10A (0.43) PDE10ATRPV3CASP3TRPV4CHEK1
SCHEMBL22042748 0.78 PDE10A (0.43) PDE10ATRPV3CASP3TRPV4CHEK1
SCHEMBL30969081 0.78 PDE10A (0.43) PDE10ATRPV3CASP3TRPV4CHEK1
SCHEMBL30151270 0.73 MAPT (0.43) KMT2AKDM4E
SCHEMBL30151235 0.71 PTGS1 (0.40) PDE10ATRPV3CASP3TRPV4PIK3CD
SCHEMBL30151240 0.71 PTGS1 (0.40) PDE10ATRPV3CASP3TRPV4PIK3CD
SCHEMBL25180910 0.71 CCR1 (0.42) PDE10AAURKAKDRAURKBKMT2A
SCHEMBL5746444 0.71 CASP3 (0.45) TRPV3CASP3TRPV4PIK3CDPIK3CA
SCHEMBL9155754 0.70 KDM4E (0.49) PDE10AKMT2ATRPV4KDM4EPIK3CA
SCHEMBL31414063 0.70 KDM4E (0.49) PDE10AKMT2ATRPV4KDM4EPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023085142-A1 FLUORINE-CONTAINING PYRIMIDINE COMPOUNDS, HARMFUL FUNGI CONTROL AGENT, AND METHOD FOR PRODUCING FLUORINE-CONTAINING PYRIMIDINE COMPOUNDS ユニマテック株式会社 2023-05-19 WO disclosed