SCHEMBL25196992

SCHEMBL25196992

O=C1CCN(C(=O)NCc2c(Cl)cccc2Cl)CC1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 6/20 0.48
KMT2A Q03164 4/20 0.45
TDP1 Q9NUW8 1/20 0.45
POLB P06746 1/20 0.44
EPHX2 P34913 2/20 0.43
LMNA P02545 2/20 0.43
HTT P42858 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
MEN1 O00255 1/20 0.43
RECQL P46063 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
PKM P14618 3/20 0.42
ALDH1A1 P00352 1/20 0.42
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25195678 0.84 PKM (0.45) P2RX7KMT2APOLBSMN1; SMN2MEN1
SCHEMBL5477278 0.82 KMT2A (0.58) P2RX7KMT2APOLBLMNAHTT
SCHEMBL25218628 0.81 NPSR1 (0.51) P2RX7KMT2AEPHX2SMN1; SMN2MEN1
SCHEMBL27196377 0.78 POLB (0.70) KMT2ATDP1POLBLMNAHTT
SCHEMBL7437717 0.78 DGAT1 (0.47) KMT2APOLBMEN1RECQLNPSR1
SCHEMBL25198233 0.77 NPC1 (0.53) P2RX7KMT2ATDP1POLBEPHX2
SCHEMBL25203080 0.75 EPHX2 (0.46) P2RX7KMT2AEPHX2MEN1NPSR1
SCHEMBL25210763 0.75 KMT2A (0.48) P2RX7KMT2ATDP1POLBMEN1
SCHEMBL5459563 0.75 ALDH1A1 (0.55) P2RX7KMT2ATDP1EPHX2LMNA
SCHEMBL25204797 0.75 P2RX7 (0.56) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023090853-A1 NOVEL UREA-BASED OR CARBAMATE-BASED P2X7 RECEPTOR ANTAGONIST, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING MAJOR DEPRESSIVE DISORDER, COMPRISING SAME AS ACTIVE INGREDIENT 고려대학교 세종산학협력단 2023-05-25 WO disclosed