SCHEMBL25201725

SCHEMBL25201725

NNc1cc(OC(F)F)ccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.44
GRM4 Q14833 2/20 0.38
TDP1 Q9NUW8 1/20 0.37
MAPT P10636 2/20 0.37
GAA P10253 1/20 0.37
ABL1 P00519 1/20 0.37
ALOX15 P16050 1/20 0.35
GFER P55789 1/20 0.35
ADAM17 P78536 1/20 0.35
GCK P35557 3/20 0.34
TSHR P16473 1/20 0.34
GSK3A P49840 2/20 0.34
GSK3B P49841 2/20 0.34
ACVR1 Q04771 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
RIOK2 Q9BVS4 1/20 0.33
TGFBR1 P36897 1/20 0.33
TGFBR2 P37173 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25211019 0.79 KDR (0.40) MAPTGAAABL1ALOX15NPC1
SCHEMBL29598523 0.76 NOS3 (0.57) ROCK1GRM4MAP4K4
SCHEMBL30001628 0.76 NOS3 (0.57) ROCK1GSK3ARIOK2
SCHEMBL17923115 0.76 NOS3 (0.57) ROCK1GRM4MAP4K4
SCHEMBL2570584 0.76 NOS3 (0.57) ROCK1GSK3ARIOK2
Hydrochloric Acid SCHEMBL25419569 0.74 NOS3 (0.55) ROCK1GSK3ARIOK2
SCHEMBL27958617 0.73 GRM4 (0.39) ROCK1GRM4TDP1MAPTABL1
SCHEMBL25229618 0.73 NOS1 (0.46) TDP1MAPTGAATSHRNPC1
SCHEMBL22658302 0.73 ROCK1 (0.42) ROCK1TDP1MAPTGAAABL1
SCHEMBL29433388 0.73 ROCK1 (0.42) ROCK1TDP1MAPTGAAABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023091726-A1 INHIBITORS OF CYCLIN‑DEPENDENT KINASE 12 (CDK12) SYROS PHARMACEUTICALS, INC. (US) 2023-05-25 WO disclosed
WO-2023091726-A1 INHIBITORS OF CYCLIN‑DEPENDENT KINASE 12 (CDK12) SYROS PHARMACEUTICALS, INC. (US) 2023-05-25 WO disclosed