SCHEMBL2521287

SCHEMBL2521287

CC(=O)NCc1cc(C2=NOC(c3cc(Cl)c(Cl)c(Cl)c3)(C(F)(F)F)C2)ccc1Br

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
F10 P00742 1/20 0.34
CA1 P00915 3/20 0.33
CA2 P00918 3/20 0.33
POLB P06746 1/20 0.33
PTPN1 P18031 1/20 0.32
PTGS2 P35354 1/20 0.32
EPHX2 P34913 1/20 0.30
NR1H4 Q96RI1 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
PDK2 Q15119 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2524229 0.92 F10 (0.35) F10CA1CA2POLBPTGS2
SCHEMBL2524696 0.90 MTOR (0.34) F10CA1CA2POLBPTGS2
SCHEMBL2515257 0.89 PDE3B (0.34) CA1CA2
SCHEMBL27893939 0.85 CA1 (0.31) CA1CA2
SCHEMBL2524706 0.85 F10 (0.34) F10CA1CA2POLBPTGS2
SCHEMBL2523120 0.85 MTOR (0.34) F10CA1CA2POLBPTGS2
SCHEMBL14234758 0.84 F10 (0.35) F10CA1CA2POLBPTGS2
SCHEMBL14685933 0.83 P2RX7 (0.32) F10CA1CA2EPHX2NR1H4
SCHEMBL2523822 0.83
SCHEMBL2522212 0.83 LMNA (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2556060-A1 SUBSTITUTED 3,5- DIPHENYL-ISOXAZOLINE DERIVATIVES AS INSECTICIDES AND ACARICIDES AH USA 42 LLC (US) 2013-02-13 EP claimed
CN-102933563-A Substituted 3,5-di phenyl-isoxazoline derivatives as insecticides and acaricides AH US 42 CO LTD 2013-02-13 CN claimed
WO-2011124998-A1 SUBSTITUTED 3,5- DI PHENYL - ISOXAZOLINE DERIVATIVES AS INSECTICIDES AND ACARICIDES PFIZER INC. (US) 2011-10-13 WO claimed
US-20110251247-A1 SUBSTITUTED ISOXAZOLINE DERIVATIVES PFIZER INC. (US) 2011-10-13 US claimed
EP-2556060-A1 SUBSTITUTED 3,5- DIPHENYL-ISOXAZOLINE DERIVATIVES AS INSECTICIDES AND ACARICIDES AH USA 42 LLC (US) 2013-02-13 EP disclosed
CN-102933563-A Substituted 3,5-di phenyl-isoxazoline derivatives as insecticides and acaricides AH US 42 CO LTD 2013-02-13 CN disclosed
WO-2011124998-A1 SUBSTITUTED 3,5- DI PHENYL - ISOXAZOLINE DERIVATIVES AS INSECTICIDES AND ACARICIDES PFIZER INC. (US) 2011-10-13 WO disclosed
WO-2011124998-A1 SUBSTITUTED 3,5- DI PHENYL - ISOXAZOLINE DERIVATIVES AS INSECTICIDES AND ACARICIDES PFIZER INC. (US) 2011-10-13 WO disclosed
US-20110251247-A1 SUBSTITUTED ISOXAZOLINE DERIVATIVES PFIZER INC. (US) 2011-10-13 US disclosed
US-20110251247-A1 SUBSTITUTED ISOXAZOLINE DERIVATIVES PFIZER INC. (US) 2011-10-13 US disclosed
US-20110251247-A1 SUBSTITUTED ISOXAZOLINE DERIVATIVES PFIZER INC. (US) 2011-10-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110251247-A1 SUBSTITUTED ISOXAZOLINE DERIVATIVES CYP4X1, COL1A1, RDX F10 1451/4885CA1 2771/4885CA2 1675/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.