SCHEMBL25237261

SCHEMBL25237261

Cc1cc(Cl)nc(Br)c1C(=O)N1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
LMNA P02545 1/20 0.45
GPR119 Q8TDV5 2/20 0.41
KCNH2 Q12809 2/20 0.41
MAPT P10636 1/20 0.40
HDAC4 P56524 1/20 0.40
PARP1 P09874 1/20 0.39
STS P08842 1/20 0.39
ACACB O00763 4/20 0.39
SPR P35270 1/20 0.39
BACE1 P56817 1/20 0.39
SCD5 Q86SK9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30496267 1.00 POLB (0.47) POLBMEN1KMT2ALMNAGPR119
SCHEMBL25874513 0.88 LMNA (0.47) POLBMEN1KMT2ALMNAGPR119
SCHEMBL25297742 0.82 ALDH1A1 (0.40) MEN1KMT2ALMNAMAPT
SCHEMBL19869973 0.81 LMNA (0.51) POLBMEN1KMT2ALMNAGPR119
SCHEMBL25738732 0.81 POLB (0.49) POLBMEN1KMT2ALMNAGPR119
SCHEMBL30478271 0.81 POLB (0.49) POLBMEN1KMT2ALMNAGPR119
SCHEMBL25238790 0.76 EHMT2 (0.48) POLBMEN1KMT2ALMNAMAPT
SCHEMBL10248751 0.75 MEN1 (0.54) POLBMEN1KMT2AGPR119MAPT
SCHEMBL19869962 0.75 LMNA (0.46) POLBMEN1KMT2ALMNASTS
SCHEMBL25738979 0.73 POLB (0.65) POLBMEN1KMT2ALMNAGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4452984-A1 DEUBIQUITINASE INHIBITORS AND METHODS OF USE THEREOF Molecure S.A. (PL) 2024-10-30 EP disclosed
US-20230219973-A1 DEUBIQUITINASE INHIBITORS AND METHODS OF USE THEREOF MOLECURE S.A. (PL) 2023-07-13 US disclosed
WO-2023119233-A1 DEUBIQUITINASE INHIBITORS AND METHODS OF USE THEREOF MOLECURE S.A. (PL) 2023-06-29 WO disclosed
WO-2023119233-A1 DEUBIQUITINASE INHIBITORS AND METHODS OF USE THEREOF MOLECURE S.A. (PL) 2023-06-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230219973-A1 DEUBIQUITINASE INHIBITORS AND METHODS OF USE THEREOF USP7, USP28, USP1 POLB 2336/4885MEN1 2177/4885KMT2A 884/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.