SCHEMBL25253418

SCHEMBL25253418

CC(Nc1cccc2c1[nH]c1ccc(-c3ccc4c(c3)CNC4=O)cc12)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TARS1 P26639 1/20 0.42
CLK4 Q9HAZ1 3/20 0.40
DYRK1B Q9Y463 2/20 0.40
TYRO3 Q06418 1/20 0.40
NTRK2 Q16620 1/20 0.40
PIM1 P11309 3/20 0.39
GSK3B P49841 2/20 0.39
DAPK3 O43293 1/20 0.39
NTRK1 P04629 1/20 0.39
FLT3 P36888 1/20 0.39
ROCK1 Q13464 1/20 0.39
PARP10 Q53GL7 1/20 0.39
PARP11 Q9NR21 1/20 0.39
TBK1 Q9UHD2 1/20 0.37
EGFR P00533 3/20 0.36
PRKCI P41743 1/20 0.36
GRM5 P41594 1/20 0.36
PRF1 P14222 2/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30455449 1.00 TARS1 (0.42) TARS1CLK4DYRK1BTYRO3NTRK2
SCHEMBL25246903 0.92 CLK4 (0.51) TARS1CLK4DYRK1BTYRO3NTRK2
SCHEMBL30455490 0.92 CLK4 (0.51) TARS1CLK4DYRK1BTYRO3NTRK2
SCHEMBL30455553 0.91 PARP11 (0.53) PIM1GSK3BPARP10PARP11EGFR
SCHEMBL25248465 0.91 PARP11 (0.53) PIM1GSK3BPARP10PARP11EGFR
SCHEMBL25247709 0.86 ROCK2 (0.34) CLK4DYRK1BTYRO3NTRK2PIM1
SCHEMBL30456104 0.86 ROCK2 (0.34) CLK4DYRK1BTYRO3NTRK2PIM1
SCHEMBL25245298 0.85 PARP10 (0.42) CLK4DYRK1BTYRO3NTRK2PIM1
SCHEMBL30455485 0.85 PARP10 (0.42) CLK4DYRK1BTYRO3NTRK2PIM1
SCHEMBL25246086 0.83 OPRD1 (0.41) EGFRPRF1PLA2G7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023121238-A1 SUBSTITUTED HETEROCYCLIC DERIVATIVE COMPOUND AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING CANCER COMPRISING SAME (주)메디픽 2023-06-29 WO claimed
WO-2023121238-A1 SUBSTITUTED HETEROCYCLIC DERIVATIVE COMPOUND AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING CANCER COMPRISING SAME (주)메디픽 2023-06-29 WO disclosed
WO-2023121238-A1 SUBSTITUTED HETEROCYCLIC DERIVATIVE COMPOUND AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING CANCER COMPRISING SAME (주)메디픽 2023-06-29 WO disclosed