SCHEMBL25256792

SCHEMBL25256792

O=C(O)/C(=C/c1ccc(O)cc1)CCc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.56
CYP2C9 P11712 1/20 0.56
AKR1B10 O60218 2/20 0.48
AKR1B1 P15121 2/20 0.48
MAOB P27338 1/20 0.48
MMP1 P03956 1/20 0.48
MMP2 P08253 1/20 0.48
MMP9 P14780 1/20 0.48
TAAR1 Q96RJ0 1/20 0.47
KEAP1 Q14145 1/20 0.47
DPP4 P27487 1/20 0.46
ALOX5 P09917 2/20 0.46
PTGES O14684 1/20 0.46
PPARG P37231 1/20 0.46
MAPT P10636 1/20 0.46
TRPV1 Q8NER1 2/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 1/20 0.44
FFAR1 O14842 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25302225 0.91 CYP3A4 (0.53) CYP3A4CYP2C9AKR1B10AKR1B1MAOB
SCHEMBL584959 0.90 CYP3A4 (0.68) CYP3A4CYP2C9KEAP1ALOX5PTGES
SCHEMBL19437149 0.90 CYP3A4 (0.68) CYP3A4CYP2C9KEAP1ALOX5PTGES
SCHEMBL19437161 0.90 CYP3A4 (0.68) CYP3A4CYP2C9KEAP1ALOX5PTGES
SCHEMBL25259728 0.86 ALOX5 (0.54) CYP3A4CYP2C9AKR1B10AKR1B1KEAP1
Water SCHEMBL29551973 0.85 CYP3A4 (0.62) CYP3A4CYP2C9KEAP1ALOX5PTGES
SCHEMBL28209668 0.83 CYP3A4 (0.80) CYP3A4CYP2C9AKR1B10AKR1B1MAOB
SCHEMBL15419989 0.83 CYP3A4 (0.80) CYP3A4CYP2C9AKR1B10AKR1B1MAOB
SCHEMBL25301706 0.83 ALDH1A1 (0.56) CYP3A4CYP2C9AKR1B10AKR1B1MMP1
SCHEMBL15263105 0.83 ALOX15 (0.52) CYP3A4CYP2C9AKR1B10AKR1B1MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3423429-B1 MODULATORS OF LIPOXYGENASE AND CYCLOOXYGENASE ENZYME ACTIVITY UNIV DE MONCTON (CA) 2023-07-12 EP claimed