SCHEMBL252676

SCHEMBL252676

C=CC[C@@H](O)CCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.45
MMP13 P45452 2/20 0.45
MMP12 P39900 2/20 0.45
MMP2 P08253 1/20 0.45
MMP9 P14780 1/20 0.45
MMP14 P50281 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.42
CYP2C19 P33261 1/20 0.42
ANPEP P15144 2/20 0.41
ERAP1 Q9NZ08 2/20 0.41
ERAP2 Q6P179 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
MAPT P10636 1/20 0.40
ACP3 P15309 1/20 0.40
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
SLC6A3 Q01959 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3904160 1.00 DPP4 (0.45) DPP4MMP13MMP12MMP2MMP9
SCHEMBL3239288 1.00 DPP4 (0.45) DPP4MMP13MMP12MMP2MMP9
SCHEMBL13841298 0.91 DPP4 (0.42) DPP4MMP13MMP12MMP2MMP9
SCHEMBL7092136 0.87 TRPA1 (0.53) MAPT
SCHEMBL9685330 0.86 TRPA1 (0.55) MAPT
SCHEMBL15944478 0.83 ESR1 (0.46) DPP4CYP2C19TDP1SLC6A2
SCHEMBL2690709 0.83 DPP4 (0.44) DPP4MMP13MMP12MMP2MMP9
SCHEMBL4799370 0.81 MMP2 (0.55) DPP4MMP13MMP12MMP2MMP9
SCHEMBL2369596 0.80 TRPA1 (0.44) SMN1; SMN2CYP2C19SLC6A2SLC6A4SLC6A3
SCHEMBL15184700 0.80 TRPA1 (0.44) SMN1; SMN2CYP2C19SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8513452-B1 Brønsted acid-catalyzed asymmetric allylation and propargylation of aldehydes UNIVERSITY OF SOUTH FLORIDA (US) 2013-08-20 US disclosed
US-8513452-B1 Brønsted acid-catalyzed asymmetric allylation and propargylation of aldehydes UNIVERSITY OF SOUTH FLORIDA (US) 2013-08-20 US disclosed
US-8088955-B2 Alpha-substituted α,β-unsaturated E- or Z-aldehydes, use thereof, and processes for their preparation α,β DSM FINE CHEMICALS AUSTRIA NFG GMBH & CO. KG (AT) 2012-01-03 US disclosed
US-20110301365-A1 ALPHA-SUBSTITUTED ALPHA, BETA-UNSATURATED E- OR Z-ALDEHYDES, USE THEREOF, AND PROCESSES FOR THEIR PREPARATION ALPHA, BETA DSM IP ASSETS B.V. (NL) 2011-12-08 US disclosed
US-20100234630-A1 ALPHA-SUBSTITUTED A,B-UNSATURATED E- OR Z-ALDEHYDES, USE THEREOF, AND PROCESSES FOR THEIR PREPARATION A,B DSM FINE CHEMICALS AUSTRIA NFG GMBH & COKG (AT) 2010-09-16 US disclosed
EP-2178816-A1 ALPHA-SUBSTITUTED , -UNSATURATED E- OR Z-ALDEHYDES, USE THEREOF, AND PROCESSES FOR THEIR PREPARATION , DSM Fine Chemicals Austria Nfg GmbH & Co KG (AT) 2010-04-28 EP disclosed
WO-2009007462-A1 ALPHA-SUBSTITUTED α,β-UNSATURATED E- OR Z-ALDEHYDES, USE THEREOF, AND PROCESSES FOR THEIR PREPARATION α,β DSM FINE CHEMICALS AUSTRIA NFG GMBH & CO. KG (AT) 2009-01-15 WO disclosed
US-4983766-A Chemical intermediates for optically active secondary alcohols IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-01-08 US disclosed
US-4812476-A SECONDARY ALCOHOLS FROM ALDEHYDE AND 3-HYDROXYBUTYRIC ACID IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-03-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110301365-A1 ALPHA-SUBSTITUTED ALPHA, BETA-UNSATURATED E- OR Z-ALDEHYDES, USE THEREOF, AND PROCESSES FOR THEIR PREPARATION ALPHA, BETA CYP8B1, ECH1, NR1H2 DPP4 3659/4885MMP13 4493/4885MMP12 3757/4885
US-20100234630-A1 ALPHA-SUBSTITUTED A,B-UNSATURATED E- OR Z-ALDEHYDES, USE THEREOF, AND PROCESSES FOR THEIR PREPARATION A,B CYP8B1, CYP1B1, ADRA1A DPP4 3912/4885MMP13 4485/4885MMP12 3943/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.