SCHEMBL25273695

SCHEMBL25273695

Nc1ccc(-c2cnnc(Cl)c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.44
TDP1 Q9NUW8 3/20 0.44
TP53 P04637 2/20 0.44
CYP3A4 P08684 2/20 0.44
HSD17B10 Q99714 4/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
KDM4E B2RXH2 3/20 0.41
MAPT P10636 3/20 0.41
HPGD P15428 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
GABRA1 P14867 2/20 0.38
GABRG2 P18507 2/20 0.38
GABRB3 P28472 2/20 0.38
GABRA5 P31644 2/20 0.38
GABRA3 P34903 2/20 0.38
TAAR1 Q96RJ0 2/20 0.38
PRKCZ Q05513 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10536955 0.83 AHR (0.41) KDM4EGABRA1GABRG2GABRB3GABRA5
SCHEMBL30530583 0.80 CYP11B2 (0.46) ALDH1A1TP53CYP3A4HSD17B10NPC1
SCHEMBL1691594 0.80 CYP11B2 (0.46) ALDH1A1TP53CYP3A4HSD17B10NPC1
SCHEMBL25220858 0.80 ESR1 (0.44) TP53NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL10535504 0.80 CYP11B2 (0.39) ALDH1A1TDP1HSD17B10NPC1RAB9A
SCHEMBL30072473 0.79 GABRG2 (0.61) ALDH1A1TDP1NPC1RAB9AKDM4E
SCHEMBL5114621 0.79 GABRG2 (0.61) ALDH1A1TDP1NPC1RAB9AKDM4E
SCHEMBL24196370 0.77 ALDH1A1 (0.38) ALDH1A1TDP1CYP3A4MEN1KMT2A
SCHEMBL4716113 0.76 TP53 (0.46) ALDH1A1TP53HSD17B10NPC1RAB9A
SCHEMBL4717600 0.76 KIF11 (0.47) ALDH1A1HSD17B10NPC1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12570650-B2 6-substituted pyridazine compounds as SMARCA2 and/or SMARCA4 degraders AURIGENE ONCOLOGY LIMITED (IN) 2026-03-10 US disclosed
US-20240018134-A1 6-Substituted Pyridazine Compounds as SMARCA2 and/or SMARCA4 Degraders AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2024-01-18 US disclosed
US-20240018134-A1 6-Substituted Pyridazine Compounds as SMARCA2 and/or SMARCA4 Degraders AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2024-01-18 US disclosed
US-20240018134-A1 6-Substituted Pyridazine Compounds as SMARCA2 and/or SMARCA4 Degraders AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2024-01-18 US disclosed
CN-116529250-A 6-substituted pyridazine compounds as SMARCA2 and/or SMARCA4 degrading agents 奥里吉恩肿瘤学有限公司 2023-08-01 CN disclosed
EP-4192835-A1 6-SUBSTITUTED PYRIDAZINE COMPOUNDS AS SMARCA2 AND/OR SMARCA4 DEGRADERS Aurigene Oncology Limited (IN) 2023-06-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240018134-A1 6-Substituted Pyridazine Compounds as SMARCA2 and/or SMARCA4 Degraders SMARCC1, SMARCC2, SMARCA4 ALDH1A1 1495/4885TDP1 244/4885TP53 412/4885
US-12570650-B2 6-substituted pyridazine compounds as SMARCA2 and/or SMARCA4 degraders SMARCC1, SMARCC2, SMARCA1 ALDH1A1 1002/4885TDP1 348/4885TP53 249/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.