SCHEMBL25289986

SCHEMBL25289986

C=CC(=O)Nc1cccc(Cl)c1C

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.61
ALDH1A1 P00352 3/20 0.56
LMNA P02545 4/20 0.54
POLB P06746 3/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
KDM4E B2RXH2 2/20 0.52
TRPV1 Q8NER1 2/20 0.52
HPGD P15428 1/20 0.52
MAPK1 P28482 1/20 0.52
TSHR P16473 1/20 0.50
HTT P42858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29410377 1.00 MAPT (0.61) MAPTALDH1A1LMNAPOLBSMN1; SMN2
SCHEMBL17931668 0.83 NPC1 (0.51) MAPTALDH1A1LMNAPOLBHPGD
SCHEMBL31162452 0.83 NPC1 (0.51) MAPTALDH1A1LMNAPOLBHPGD
SCHEMBL2093176 0.82 MAPT (0.69) MAPTALDH1A1LMNAPOLBSMN1; SMN2
SCHEMBL10477308 0.82 MMP1 (0.60) MAPTLMNAKDM4EHPGD
SCHEMBL30452125 0.82 MMP1 (0.60) MAPTLMNAKDM4EHPGD
SCHEMBL7191119 0.81 BTK (0.49) MAPTALDH1A1LMNAPOLBTRPV1
SCHEMBL8512135 0.81 MMP1 (0.58) KDM4EHPGD
SCHEMBL6474649 0.81 MAPT (0.67) MAPTALDH1A1LMNAPOLBSMN1; SMN2
SCHEMBL952943 0.81 MAPT (0.58) MAPTALDH1A1LMNAPOLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117466789-A Synthesis method of beta-trifluoromethylthioamide participated by silver trifluormethane 陕西先氟领创科技有限公司 2024-01-30 CN claimed
US-12630516-B2 Compounds NRG THERAPEUTICS LTD. (GB) 2026-05-19 US disclosed
US-12497359-B2 Acrylamide derivatives NRG THERAPEUTICS LTD (GB) 2025-12-16 US disclosed
EP-4208442-B1 MPTP INHIBITORS NRG THERAPEUTICS LTD (GB) 2025-10-22 EP disclosed
US-20250179028-A1 ACRYLAMIDE COMPOUNDS NRG THERAPEUTICS LTD (GB) 2025-06-05 US disclosed
EP-4208448-B1 ACRYLAMIDE DERIVATIVES NRG THERAPEUTICS LTD (GB) 2025-04-23 EP disclosed
EP-4486721-A1 ACRYLAMIDE COMPOUNDS NRG Therapeutics LTD (GB) 2025-01-08 EP disclosed
US-20240067614-A1 NOVEL COMPOUNDS NRG THERAPEUTICS LTD. (GB) 2024-02-29 US disclosed
US-20240067614-A1 NOVEL COMPOUNDS NRG THERAPEUTICS LTD. (GB) 2024-02-29 US disclosed
US-20240067614-A1 NOVEL COMPOUNDS NRG THERAPEUTICS LTD. (GB) 2024-02-29 US disclosed
US-20230312466-A1 NOVEL COMPOUNDS NRG THERAPEUTICS LTD (GB) 2023-10-05 US disclosed
US-20230312466-A1 NOVEL COMPOUNDS NRG THERAPEUTICS LTD (GB) 2023-10-05 US disclosed
WO-2023166303-A1 ACRYLAMIDE COMPOUNDS NRG THERAPEUTICS LTD (GB) 2023-09-07 WO disclosed
WO-2023166303-A1 ACRYLAMIDE COMPOUNDS NRG THERAPEUTICS LTD (GB) 2023-09-07 WO disclosed
EP-4208442-A1 NOVEL COMPOUNDS NRG Therapeutics LTD (GB) 2023-07-12 EP disclosed
EP-4208448-A1 NOVEL COMPOUNDS NRG Therapeutics LTD (GB) 2023-07-12 EP disclosed
CN-116096705-A Novel compounds NRG治疗有限公司 2023-05-09 CN disclosed
CN-116096712-A Novel compounds NRG治疗有限公司 2023-05-09 CN disclosed
WO-2022049376-A1 NOVEL COMPOUNDS NRG THERAPEUTICS LTD (GB) 2022-03-10 WO disclosed
WO-2022049377-A1 NOVEL COMPOUNDS NRG THERAPEUTICS LTD (GB) 2022-03-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12630516-B2 Compounds CYP4B1, CYP1B1, NR4A1 MAPT 2453/4885ALDH1A1 87/4885LMNA 1708/4885
US-20230312466-A1 NOVEL COMPOUNDS CYP11B1, CYP11B2, UGT1A1 MAPT 2537/4885ALDH1A1 516/4885LMNA 3307/4885
US-20240067614-A1 NOVEL COMPOUNDS CYP11B1, CYP11B2, CXCR2 MAPT 2596/4885ALDH1A1 478/4885LMNA 3273/4885
US-20250179028-A1 ACRYLAMIDE COMPOUNDS ACR, CCNI, FANCI MAPT 1371/4885ALDH1A1 63/4885LMNA 1086/4885
US-12497359-B2 Acrylamide derivatives ACR, GSTA2, GSTA1 MAPT 1784/4885ALDH1A1 48/4885LMNA 1162/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.