SCHEMBL252900

SCHEMBL252900

C=CCC(Cc1ccccc1)C(=O)O

nearest known ligand 0.68

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.68
CPA1 P15085 7/20 0.59
CPA3 P15088 3/20 0.59
FOLH1 Q04609 3/20 0.59
CPB1 P15086 1/20 0.59
CPB2 Q96IY4 1/20 0.59
MME P08473 3/20 0.56
SLC1A3 P43003 1/20 0.54
SLC1A2 P43004 1/20 0.54
SLC1A1 P43005 1/20 0.54
CYP2C19 P33261 1/20 0.53
NAALAD2 Q9Y3Q0 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL629350 1.00 CYP1A2 (0.68) CYP1A2CPA1CPA3FOLH1CPB1
SCHEMBL9007628 1.00 CYP1A2 (0.68) CYP1A2CPA1CPA3FOLH1CPB1
SCHEMBL5096045 0.86 PTGS2 (0.51) CYP1A2CPA1CPA3FOLH1CPB1
SCHEMBL11324047 0.86 CYP1A2 (0.53) CYP1A2CPA1CPA3FOLH1CPB1
SCHEMBL2065619 0.86 CYP1A2 (0.53) CYP1A2CPA1CPA3FOLH1CPB1
SCHEMBL2361534 0.86 CYP1A2 (0.53) CYP1A2CPA1CPA3FOLH1CPB1
SCHEMBL8144720 0.86 CYP1A2 (0.53) CYP1A2CPA1CPA3FOLH1CPB1
SCHEMBL5966473 0.85 PPARG (0.58) CYP1A2
SCHEMBL9647546 0.85 SLC1A1 (0.77) CYP1A2SLC1A3SLC1A2SLC1A1
SCHEMBL8301284 0.84 PPARG (0.48) CYP1A2CPA1CPA3MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 52 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832923-A1 Polyamide-acrylonitrile butadiene blends with reduced gel and antigel agent THE GOODYEAR TIRE & RUBBER COMPANY (US) 1998-04-01 EP claimed
EP-0192492-B1 PEPTIDES CONTAINING AN ALIPHATIC-AROMATIC KETONE SIDE CHAIN THE SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 1992-01-02 EP claimed
US-20160046590-A1 SONIC HEDGEHOG MODULATORS MASSACHUSETTS INST TECHNOLOGY (US) 2016-02-18 US disclosed
US-8530456-B2 Sonic hedgehog modulators PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2013-09-10 US disclosed
US-8470763-B2 Alpha-amino-N-substituted amides, pharmaceutical composition containing them and uses thereof SHANGHAI INSTITUTE OF MATERIA MEDICA CHINESE ACADEMY OF SCIENCES (CN) 2013-06-25 US disclosed
US-8470763-B2 Alpha-amino-N-substituted amides, pharmaceutical composition containing them and uses thereof SHANGHAI INSTITUTE OF MATERIA MEDICA CHINESE ACADEMY OF SCIENCES (CN) 2013-06-25 US disclosed
EP-1948643-B1 3-ALKYL-5- (4-ALKYL-5-OXO-TETRAHYDROFURAN-2-YL) PYRROLIDIN-2-ONE DERIVATIVES AS INTERMEDIATES IN THE SYNTHESIS OF RENIN INHIBITORS NOVARTIS AG (CH) 2013-06-05 EP disclosed
US-8338620-B2 Methods for the production of C-8 lactam lactone compounds NOVARTIS AG (CH) 2012-12-25 US disclosed
US-8198465-B2 3-alkyl-5- (4-alkyl-5-oxo-tetrahydrofutran-2-yl) pyrrolidin-2-one derivatives as intermediates in the synthesis of renin inhibitors NOVARTIS AG (CH) 2012-06-12 US disclosed
EP-1296927-B1 PREPARATION OF (R)-2-ALKYL-3-PHENYLPROPIONIC ACIDS NOVARTIS AG (CH) 2012-02-22 EP disclosed
US-8088955-B2 Alpha-substituted α,β-unsaturated E- or Z-aldehydes, use thereof, and processes for their preparation α,β DSM FINE CHEMICALS AUSTRIA NFG GMBH & CO. KG (AT) 2012-01-03 US disclosed
US-20030139625-A1 Preparation of (r -2-alkyl-3-phenylpropionic acids SPEEDEL PHARMA AG (CH) 2003-07-24 US disclosed
EP-1296912-A1 PROCESS FOR THE PREPARATION OF (R)-2-ALKYL-3-PHENYL-1-PROPANOLS Speedel Pharma AG (CH) 2003-04-02 EP disclosed
EP-1296927-A1 PREPARATION OF (R)-2-ALKYL-3-PHENYLPROPIONIC ACIDS Speedel Pharma AG (CH) 2003-04-02 EP disclosed
WO-2002002500-A1 PREPARATION OF (R)-2-ALKYL-3-PHENYLPROPIONIC ACIDS SPEEDEL PHARMA AG (CH) 2002-01-10 WO disclosed
WO-2002002487-A1 PROCESS FOR THE PREPARATION OF (R)-2-ALKYL-3-PHENYL-1-PROPANOLS SPEEDEL PHARMA AG (CH) 2002-01-10 WO disclosed
US-5852086-A Polyamide-acrylonitrile butadiene blends with reduced gel and antigel agent THE GOODYEAR TIRE & RUBBER COMPANY (US) 1998-12-22 US disclosed
EP-0832923-A1 Polyamide-acrylonitrile butadiene blends with reduced gel and antigel agent THE GOODYEAR TIRE & RUBBER COMPANY (US) 1998-04-01 EP disclosed
US-5569762-A Asymmetric synthesis of intermediates for retroviral protease inhibitor compounds AMERICAN CYANAMID COMPANY (US) 1996-10-29 US disclosed
US-5428167-A Asymmetric synthesis of intermediates for retroviral protease inhibitor compounds AMERICAN CYANAMID COMPANY (US) 1995-06-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030139625-A1 Preparation of (r -2-alkyl-3-phenylpropionic acids PCCA, APEH, ALDH1A1 CYP1A2 141/4885CPA1 72/4885CPA3 221/4885
US-20160046590-A1 SONIC HEDGEHOG MODULATORS SHH, GLI1, SMO CYP1A2 4873/4885CPA1 3702/4885CPA3 4092/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.