SCHEMBL2530643

SCHEMBL2530643

CC(C(=O)O)C1NC(=O)c2cc(O)ccc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.37
ESR2 Q92731 3/20 0.37
MAOA P21397 1/20 0.37
UGT1A1 P22309 1/20 0.37
MAOB P27338 1/20 0.37
ANPEP P15144 1/20 0.37
DPP4 P27487 1/20 0.37
LMNA P02545 2/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
RECQL P46063 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TTR P02766 1/20 0.33
KMT2A Q03164 2/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
MEN1 O00255 1/20 0.32
HIF1A Q16665 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18209300 0.87 EDNRB (0.42) KMT2AMEN1
SCHEMBL18209322 0.80 HSD17B10 (0.49) LMNAMAPTSMN1; SMN2KDM4E
SCHEMBL2525409 0.73 HSD17B10 (0.48) ESR1ESR2MAOAUGT1A1MAOB
SCHEMBL18215445 0.72 EDNRB (0.44) KMT2AMEN1
SCHEMBL2522963 0.71 HSD17B1 (0.41) ESR1ESR2MAOAUGT1A1MAOB
SCHEMBL23784644 0.69 TGM2 (0.36)
SCHEMBL12214779 0.69 CYP1A2 (0.51) ESR1ESR2GAAKMT2AKDM4E
SCHEMBL17711719 0.66 MKNK1 (0.43) LMNAGAAMAPTKMT2AKDM4E
SCHEMBL6451059 0.65 TYR (0.47) LMNAGAAMAPTSMN1; SMN2NPSR1
SCHEMBL6451064 0.65 TYR (0.47) LMNAGAAMAPTSMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8039484-B2 Antidiabetic bicyclic compounds MERCK SHARP & DOHME CORP. (US) 2011-10-18 US disclosed