SCHEMBL253171

SCHEMBL253171

CCOC(=O)NNC(N)=S

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.46
ALDH1A1 P00352 5/20 0.43
HPGD P15428 2/20 0.43
HSD17B10 Q99714 2/20 0.43
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GAA P10253 2/20 0.43
MGAM O43451 1/20 0.41
SI P14410 1/20 0.41
MGAM2 Q2M2H8 1/20 0.41
KMT2A Q03164 1/20 0.38
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
SOAT1 P35610 1/20 0.36
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL32131 0.84 ALOX15 (0.52) ALOX15ALDH1A1HSD17B10LMNASMN1; SMN2
SCHEMBL355253 0.83 GAA (0.55) ALOX15ALDH1A1HSD17B10LMNASMN1; SMN2
SCHEMBL27537856 0.81 GAA (0.48) ALDH1A1HSD17B10LMNASMN1; SMN2GAA
SCHEMBL4991475 0.80 GAA (0.48) ALOX15ALDH1A1HPGDHSD17B10LMNA
SCHEMBL1233113 0.80
SCHEMBL3701771 0.80 LMNA (0.44) ALOX15ALDH1A1HSD17B10LMNASMN1; SMN2
SCHEMBL5400363 0.78 ALOX15 (0.46) ALOX15ALDH1A1HPGDHSD17B10LMNA
SCHEMBL29054143 0.78 ALOX15 (0.46) ALOX15ALDH1A1HSD17B10LMNASMN1; SMN2
SCHEMBL10818731 0.78 ALOX15 (0.46) ALOX15ALDH1A1HSD17B10LMNASMN1; SMN2
SCHEMBL689234 0.78 GAA (0.52) ALOX15ALDH1A1HPGDHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 226 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4396630-A1 ELECTROACTIVE OPTICAL DEVICE PPG Industries Ohio Inc. (US) 2024-07-10 EP claimed
EP-4347683-A1 CURABLE PHOTOCHROMIC COMPOSITION Transitions Optical, Ltd. (IE) 2024-04-10 EP claimed
US-20230416609-A1 Method for Preparing a Coated Article TRANSITIONS OPTICAL, LTD. (IE) 2023-12-28 US claimed
US-20230400616-A1 Photochromic-Dichroic Articles TRANSITIONS OPTICAL, LTD. (IE) 2023-12-14 US claimed
EP-4244304-A1 METHOD FOR PREPARING A COATED ARTICLE Transitions Optical, Ltd. (IE) 2023-09-20 EP claimed
EP-4244305-A1 PHOTOCHROMIC-DICHROIC ARTICLES Transitions Optical, Ltd. (IE) 2023-09-20 EP claimed
US-20230087427-A1 CURABLE COMPOSITIONS PPG INDUSTRIES OHIO, INC. (US) 2023-03-23 US claimed
WO-2023034737-A1 ELECTROACTIVE OPTICAL DEVICE PPG INDUSTRIES OHIO, INC. (US) 2023-03-09 WO claimed
EP-4022366-A1 PHOTOCHROMIC FILM LAMINATE Transitions Optical, Ltd. (IE) 2022-07-06 EP claimed
EP-2959340-B1 MULTI LAYER OPTICAL DEVICE TRANSITIONS OPTICAL INC (US) 2022-06-29 EP claimed
JP-2009545018-A 2009-12-17 JP claimed
US-20090309076-A1 PHOTOCHROMIC COMPOUNDS TRANSITIONS OPTICAL, INC. (US) 2009-12-17 US claimed
US-20090135462-A1 CLEAR TO CIRCULAR POLARIZING PHOTOCHROMIC DEVICES AND METHODS OF MAKING THE SAME TRANSITIONS OPTICAL, INC. (US) 2009-05-28 US claimed
EP-2047305-A1 ORIENTED POLYMERIC SHEETS EXHIBITING DICHROISM AND ARTICLES CONTAINING THE SAME TRANSITIONS OPTICAL, INC. (US) 2009-04-15 EP claimed
EP-2001966-A1 ABRASION RESISTANT COATING COMPOSITIONS AND COATED ARTICLES PPG Industries Ohio, Inc. (US) 2008-12-17 EP claimed
WO-2008111995-A1 ORIENTED POLYMERIC SHEETS EXHIBITING DICHROISM AND ARTICLES CONTAINING THE SAME TRANSITIONS OPTICAL, INC. (US) 2008-09-18 WO claimed
US-20080187749-A1 OPTICAL ELEMENT HAVING LIGHT INFLUENCING PROPERTY PPG INDUSTRIES OHIO, INC. (US) 2008-08-07 US claimed
WO-2008088633-A1 OPTICAL ELEMENT HAVING LIGHT INFLUENCING PROPERTY PPG INDUSTRIES OHIO, INC. (US) 2008-07-24 WO claimed
US-20070291345-A1 ORIENTED POLYMERIC SHEETS EXHIBITING DICHROISM AND ARTICLES CONTAINING THE SAME TRANSITIONS OPTICAL, INC. (US) 2007-12-20 US claimed
WO-2007118024-A1 ABRASION RESISTANT COATING COMPOSITIONS AND COATED ARTICLES PPG INDUSTRIES OHIO, INC. (US) 2007-10-18 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090309076-A1 PHOTOCHROMIC COMPOUNDS CCR4, CCR8, CBR3 ALOX15 1297/4885ALDH1A1 1782/4885HPGD 2895/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.