SCHEMBL25319219

SCHEMBL25319219

COC1CN(C(=O)c2ccc(NC(=O)OC(C)(C)C)nn2)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.38
GRM5 P41594 1/20 0.37
CFTR P13569 2/20 0.36
CCNC P24863 2/20 0.36
CDK8 P49336 2/20 0.36
SCN9A Q15858 1/20 0.36
GRIN2B Q13224 1/20 0.36
BCL2 P10415 1/20 0.35
GSK3B P49841 1/20 0.35
DYRK1A Q13627 1/20 0.35
RORC P51449 1/20 0.34
CDK19 Q9BWU1 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
BACE1 P56817 1/20 0.34
ATR Q13535 2/20 0.33
PDK2 Q15119 1/20 0.33
PTPN2 P17706 1/20 0.33
PTPN1 P18031 1/20 0.33
PTPN6 P29350 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31150452 1.00 GABRA1 (0.38) GABRA1GRM5CFTRCCNCCDK8
SCHEMBL29311708 0.76 GLS (0.40) GRIN2BGSK3BDYRK1A
SCHEMBL7240100 0.76 CYP17A1 (0.38) SCN9AGRIN2BBCL2GSK3BDYRK1A
SCHEMBL26839479 0.76 GSK3B (0.39) SCN9ABCL2GSK3BDYRK1AATR
SCHEMBL30565562 0.76 CYP17A1 (0.38) SCN9AGRIN2BBCL2GSK3BDYRK1A
SCHEMBL25317444 0.73 GABRA1 (0.44) GABRA1CCNCCDK8SCN9ACDK19
SCHEMBL30986515 0.71 CYP17A1 (0.36) SCN9AGRIN2BGSK3BDYRK1AATR
SCHEMBL8162669 0.70 CYP1A2 (0.42) ATR
SCHEMBL29442854 0.70 LMNA (0.53) GSK3BDYRK1AATR
SCHEMBL15202941 0.70 LMNA (0.53) GSK3BDYRK1AATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4466258-A1 NEW BENZIMIDAZOLE PYRIDINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2024-11-27 EP disclosed
WO-2023139085-A1 NEW BENZIMIDAZOLE PYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2023-07-27 WO disclosed